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2G01

Pyrazoloquinolones as Novel, Selective JNK1 inhibitors

エンティティ
Entity ID鎖名説明種類鎖長化学式量分子数データベース名(アクセス番号)由来する生物種エンティティの一般名
1A, BMitogen-activated protein kinase 8polymer37042919.62UniProt (P45983)
Pfam (PF00069)
In PDB
Homo sapiens (human)Stress-activated protein kinase JNK1, c-Jun N-terminal kinase 1, JNK-46
2F, GC-jun-amino-terminal kinase-interacting protein 1polymer111345.62UniProt (Q9UQF2)
In PDB
JNK-interacting protein 1, JIP-1, JNK MAP kinase scaffold protein 1, Islet-brain-1, IB-1, Mitogen-activated protein kinase 8-interacting protein 1
3A, BSULFATE IONnon-polymer96.14Chemie (SO4)
4A, B6-CHLORO-9-HYDROXY-1,3-DIMETHYL-1,9-DIHYDRO-4H-PYRAZOLO[3,4-B]QUINOLIN-4-ONEnon-polymer263.72Chemie (73Q)
配列変更
A, B: 1 - 364 (UniProt: P45983)
PDB外部データベース詳細
Glu 183Thr 183engineered mutation
Glu 185Tyr 185engineered mutation
His 365-expression tag
His 366-expression tag
His 367-expression tag
His 368-expression tag
His 369-expression tag
His 370-expression tag
配列ビューア
非対称単位の内容
タンパク質・
核酸鎖
鎖の数4
化学式量合計88530.3
タンパク質・
核酸・
糖鎖以外*
分子数6
化学式量合計911.6
全て*化学式量合計89442.0
*水分子は含んでいません

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件を2024-09-18に公開中

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