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1G65

Crystal structure of epoxomicin:20s proteasome reveals a molecular basis for selectivity of alpha,beta-epoxyketone proteasome inhibitors

エンティティ
Entity ID鎖名説明種類鎖長化学式量分子数データベース名(アクセス番号)由来する生物種エンティティの一般名
1A, OProteasome component Y7polymer25027191.82UniProt (P23639)
Pfam (PF10584)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit Y7, Multicatalytic endopeptidase complex subunit Y7, Proteinase YSCE subunit 7
2B, PProteasome component Y13polymer24427050.42UniProt (P23638)
Pfam (PF10584)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit Y13, Multicatalytic endopeptidase complex subunit Y13, Proteinase YSCE subunit 13
3C, QProteasome component PRE6polymer24126903.32UniProt (P40303)
Pfam (PF10584)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PRE6, Multicatalytic endopeptidase complex subunit PRE6, Proteinase YSCE subunit PRE6
4D, RProteasome component PUP2polymer24226544.82UniProt (P32379)
Pfam (PF00227)
Pfam (PF10584)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PUP2, Multicatalytic endopeptidase complex subunit PUP2, Proteinase YSCE subunit PUP2
5E, SProteasome component PRE5polymer23325502.82UniProt (P40302)
Pfam (PF10584)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PRE5, Multicatalytic endopeptidase complex subunit PRE5, Proteinase YSCE subunit PRE5
6F, TProteasome component C1polymer24426892.52UniProt (P21242)
Pfam (PF10584)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit C1, Multicatalytic endopeptidase complex subunit C1, Proteinase YSCE subunit 1
7G, UProteasome component C7-alphapolymer24327316.02UniProt (P21243)
Pfam (PF10584)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit C7-alpha, Multicatalytic endopeptidase complex C7, Proteasome component Y8, Proteinase YSCE subunit 7, SCL1 suppressor protein
8H, VProteasome component PUP1polymer22223987.32UniProt (P25043)
Pfam (PF00227)
Pfam (PF12465)
In PDB
Saccharomyces cerevisiae S288c (Baker's yeast)Macropain subunit PUP1, Multicatalytic endopeptidase complex subunit PUP1, Proteinase YSCE subunit PUP1
9I, WProteasome component PUP3polymer20422496.62UniProt (P25451)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PUP3, Multicatalytic endopeptidase complex subunit PUP3
10J, XProteasome component C11polymer19822545.72UniProt (P22141)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit C11, Multicatalytic endopeptidase complex subunit C11, Proteinase YSCE subunit 11
11K, YProteasome component PRE2polymer21223325.22UniProt (P30656)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PRE2, Multicatalytic endopeptidase complex subunit PRE2, Proteinase YSCE subunit PRE2
12L, ZProteasome component C5polymer22224883.92UniProt (P23724)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Multicatalytic endopeptidase complex subunit C5
13M, 1Proteasome component PRE4polymer23325945.52UniProt (P30657)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PRE4, Multicatalytic endopeptidase complex subunit PRE4, Proteinase YSCE subunit PRE4
14N, 2Proteasome component PRE3polymer19621517.22UniProt (P38624)
Pfam (PF00227)
In PDB
Saccharomyces cerevisiae (Baker's yeast)Macropain subunit PRE3, Multicatalytic endopeptidase complex subunit PRE3, Proteinase YSCE subunit PRE3
153, 4EPOXOMICIN (peptide inhibitor)polymer5542.82
16D, F, G, H, I...MAGNESIUM IONnon-polymer24.310Chemie (MG)
17waterwater18.02872Chemie (HOH)
配列ビューア
非対称単位の内容
タンパク質・
核酸鎖
鎖の数30
化学式量合計705291.7
タンパク質・
核酸・
糖鎖以外*
分子数10
化学式量合計243.1
全て*化学式量合計705534.8
*水分子は含んでいません

225158

件を2024-09-18に公開中

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