Summary
Title: | CDK2 in complex with a disubstituted 4, 6-bis anilino pyrimidine CDK4 inhibitor |
Citation: | Beattie, J.F.,Breault, G.A.,Ellston, R.P.A.,Green, S.,Jewsbury, P.J.,Midgley, C.J.,Naven, R.T.,Minshull, C.A.,Pauptit, R.A.,Tucker, J.A.,Pease, J.E. Cyclin-Dependent Kinase 4 Inhibitors as a Treatment for Cancer. Part 1: Identification and Optimisation of Substituted 4,6-Bis Anilino Pyrimidines Bioorg.Med.Chem.Lett., 13:2955-, 2003 |
Experimental method: | X-RAY DIFFRACTION (2.31 Å) |
Deposition date: | 2002-06-11 |
Release date: | 2003-07-11 |
Obsoletion date: | 2004-05-04 |
Timeline
Downloads
File format | File name (file size) | ||
PDBx/mmCIF | 1h06.cif.gz Display(67.48 KB) 1h06.cif | ||
PDBx/mmJSON | no-atom | 1h06-noatom.json.gz Display (Header)(10.47 KB) 1h06-noatom.json | |
PDBML | all | 1h06.xml.gz Display(89.86 KB) 1h06.xml | |
PDB | pdb1h06.ent.gz Display(54.68 KB) pdb1h06.ent | ||
Structure factors | r1h06sf.ent.gz Display(126.32 KB) r1h06sf.ent |