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6BKW

BTK complex with compound 12

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004672molecular_functionprotein kinase activity
A0004713molecular_functionprotein tyrosine kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
PDBデータベースに由来する情報
site_idAC1
残基数6
詳細binding site for residue SO4 A 701
鎖名残基
ALYS466
AARG487
AARG490
ALYS595
AHOH816
AHOH870

site_idAC2
残基数8
詳細binding site for residue SO4 A 702
鎖名残基
APRO619
AHIS620
AHOH814
AHOH847
AHOH882
ASER592
ALYS595
ATYR617

site_idAC3
残基数4
詳細binding site for residue SO4 A 703
鎖名残基
AARG490
AHIS491
ALYS637
AHOH819

site_idAC4
残基数21
詳細binding site for residue DXM A 704
鎖名残基
ALEU408
ATHR410
AGLY411
APHE413
AVAL416
AALA428
ALYS430
ATHR474
AGLU475
ATYR476
AMET477
AALA478
AGLY480
AASN526
ALEU528
AASP539
ATYR551
AHOH806
AHOH843
AHOH896
AHOH930

site_idAC5
残基数11
詳細binding site for residue FPZ A 705
鎖名残基
ATRP395
ATRP421
ATYR425
AASP426
ATYR461
ATYR598
ALEU614
AARG615
ALEU616
ATYR617
AHOH829

site_idAC6
残基数3
詳細binding site for residue GOL A 706
鎖名残基
ATYR418
ATYR476
AHOH820

site_idAC7
残基数4
詳細binding site for residue GOL A 707
鎖名残基
AARG618
AHIS620
ALEU621
AALA622

UniProtにおけるモチーフ・データベースPROSITEからの機能情報
site_idPS00107
残基数23
詳細PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. LGTGQFGVVKyGkwrgqyd...........VAIK
鎖名残基詳細
ALEU408-LYS430

site_idPS00109
残基数13
詳細PROTEIN_KINASE_TYR Tyrosine protein kinases specific active-site signature. FLHrDLAARNCLV
鎖名残基詳細
APHE517-VAL529

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数1
詳細ACT_SITE: Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10028
鎖名残基詳細
AASP521

site_idSWS_FT_FI2
残基数2
詳細BINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
鎖名残基詳細
ALEU408
ALYS430

site_idSWS_FT_FI3
残基数1
詳細BINDING: BINDING => ECO:0000269|PubMed:20052711, ECO:0007744|PDB:3K54, ECO:0007744|PDB:3OCT
鎖名残基詳細
ATHR474

site_idSWS_FT_FI4
残基数1
詳細BINDING: BINDING => ECO:0000269|PubMed:21280133, ECO:0007744|PDB:3PIY
鎖名残基詳細
ALEU542

site_idSWS_FT_FI5
残基数1
詳細MOD_RES: Phosphotyrosine; by LYN and SYK => ECO:0000269|PubMed:8630736, ECO:0000269|PubMed:9012831
鎖名残基詳細
ATYR551

site_idSWS_FT_FI6
残基数1
詳細MOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
鎖名残基詳細
ASER604

site_idSWS_FT_FI7
残基数1
詳細MOD_RES: Phosphotyrosine => ECO:0000269|PubMed:15375214
鎖名残基詳細
ATYR617

site_idSWS_FT_FI8
残基数1
詳細MOD_RES: Phosphoserine => ECO:0000269|PubMed:15375214
鎖名残基詳細
ASER623

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件を2024-09-18に公開中

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