5ZNI
Plasmodium falciparum purine nucleoside phosphorylase in complex with mefloquine
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003824 | molecular_function | catalytic activity |
A | 0004731 | molecular_function | purine-nucleoside phosphorylase activity |
A | 0004850 | molecular_function | uridine phosphorylase activity |
A | 0005829 | cellular_component | cytosol |
A | 0006166 | biological_process | purine ribonucleoside salvage |
A | 0006218 | biological_process | uridine catabolic process |
A | 0009116 | biological_process | nucleoside metabolic process |
A | 0016757 | molecular_function | glycosyltransferase activity |
A | 0047975 | molecular_function | guanosine phosphorylase activity |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 10 |
Details | binding site for residue PO4 A 301 |
Chain | Residue |
A | GLY23 |
A | HOH427 |
A | ARG27 |
A | ARG45 |
A | ARG88 |
A | GLY90 |
A | SER91 |
A | YMZ302 |
A | HOH409 |
A | HOH410 |
site_id | AC2 |
Number of Residues | 15 |
Details | binding site for residue YMZ A 302 |
Chain | Residue |
A | HIS7 |
A | ARG45 |
A | CYS92 |
A | GLY93 |
A | TYR160 |
A | VAL181 |
A | GLU182 |
A | MET183 |
A | ASP206 |
A | GLY207 |
A | CYS208 |
A | PRO209 |
A | PO4301 |
A | HOH401 |
A | HOH442 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | ACT_SITE: Proton donor => ECO:0000250|UniProtKB:Q8I3X4 |
Chain | Residue | Details |
A | ASP206 |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | BINDING: BINDING => ECO:0000250|UniProtKB:Q8I3X4 |
Chain | Residue | Details |
A | HIS7 | |
A | ARG45 |
site_id | SWS_FT_FI3 |
Number of Residues | 1 |
Details | BINDING: in other chain => ECO:0000269|PubMed:30602534, ECO:0007744|PDB:5ZNI |
Chain | Residue | Details |
A | GLY23 |
site_id | SWS_FT_FI4 |
Number of Residues | 1 |
Details | BINDING: in other chain => ECO:0000269|PubMed:30602534, ECO:0007744|PDB:5ZNC, ECO:0007744|PDB:5ZNI |
Chain | Residue | Details |
A | ARG88 |
site_id | SWS_FT_FI5 |
Number of Residues | 1 |
Details | BINDING: in other chain => ECO:0000250|UniProtKB:Q8I3X4 |
Chain | Residue | Details |
A | MET183 |