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3SKE

I. Novel HCV NS5B Polymerase Inhibitors: Discovery of Indole 2- Carboxylic Acids with C3-Heterocycles

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
PDBデータベースに由来する情報
site_idAC1
残基数9
詳細BINDING SITE FOR RESIDUE PO4 A 577
鎖名残基
APRO265
AARG505
AVAL530
AARG531
ATHR532
AHOH662
AHOH854
AHOH951
AHOH970

site_idAC2
残基数18
詳細BINDING SITE FOR RESIDUE 054 A 578
鎖名残基
APRO197
AASN316
ACYS366
ASER368
ALEU384
ASER407
AGLY410
AASN411
AMET414
ATYR415
AGLN446
AILE447
ATYR448
AHOH624
AHOH700
AHOH728
AHOH915
AHOH944

site_idAC3
残基数17
詳細BINDING SITE FOR RESIDUE 054 B 577
鎖名残基
BPRO197
BASN316
BCYS366
BSER368
BLEU384
BSER407
BGLY410
BASN411
BMET414
BTYR415
BGLN446
BILE447
BTYR448
BHOH643
BHOH727
BHOH750
BHOH848

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数6
詳細BINDING: BINDING => ECO:0000250|UniProtKB:P26663
鎖名残基詳細
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
残基数4
詳細MOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
鎖名残基詳細
ASER29
ASER42
BSER29
BSER42

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件を2024-09-18に公開中

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