3SKE
I. Novel HCV NS5B Polymerase Inhibitors: Discovery of Indole 2- Carboxylic Acids with C3-Heterocycles
GO(遺伝子オントロジー)由来の情報
鎖名 | GO(遺伝子オントロジー)id | 名前空間 | 内容 |
A | 0003723 | molecular_function | RNA binding |
A | 0003968 | molecular_function | RNA-dependent RNA polymerase activity |
A | 0039694 | biological_process | viral RNA genome replication |
B | 0003723 | molecular_function | RNA binding |
B | 0003968 | molecular_function | RNA-dependent RNA polymerase activity |
B | 0039694 | biological_process | viral RNA genome replication |
PDBデータベースに由来する情報
site_id | AC1 |
残基数 | 9 |
詳細 | BINDING SITE FOR RESIDUE PO4 A 577 |
鎖名 | 残基 |
A | PRO265 |
A | ARG505 |
A | VAL530 |
A | ARG531 |
A | THR532 |
A | HOH662 |
A | HOH854 |
A | HOH951 |
A | HOH970 |
site_id | AC2 |
残基数 | 18 |
詳細 | BINDING SITE FOR RESIDUE 054 A 578 |
鎖名 | 残基 |
A | PRO197 |
A | ASN316 |
A | CYS366 |
A | SER368 |
A | LEU384 |
A | SER407 |
A | GLY410 |
A | ASN411 |
A | MET414 |
A | TYR415 |
A | GLN446 |
A | ILE447 |
A | TYR448 |
A | HOH624 |
A | HOH700 |
A | HOH728 |
A | HOH915 |
A | HOH944 |
site_id | AC3 |
残基数 | 17 |
詳細 | BINDING SITE FOR RESIDUE 054 B 577 |
鎖名 | 残基 |
B | PRO197 |
B | ASN316 |
B | CYS366 |
B | SER368 |
B | LEU384 |
B | SER407 |
B | GLY410 |
B | ASN411 |
B | MET414 |
B | TYR415 |
B | GLN446 |
B | ILE447 |
B | TYR448 |
B | HOH643 |
B | HOH727 |
B | HOH750 |
B | HOH848 |
SwissProt/UniProtに記載されている蛋白質分子機能情報
site_id | SWS_FT_FI1 |
残基数 | 6 |
詳細 | BINDING: BINDING => ECO:0000250|UniProtKB:P26663 |
鎖名 | 残基 | 詳細 |
A | ASP220 | |
A | ASP318 | |
A | ASP319 | |
B | ASP220 | |
B | ASP318 | |
B | ASP319 |
site_id | SWS_FT_FI2 |
残基数 | 4 |
詳細 | MOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662 |
鎖名 | 残基 | 詳細 |
A | SER29 | |
A | SER42 | |
B | SER29 | |
B | SER42 |