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1T3R

HIV protease wild-type in complex with TMC114 inhibitor

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
PDBデータベースに由来する情報
site_idAC1
残基数10
詳細BINDING SITE FOR RESIDUE PO4 B 501
鎖名残基
AARG14
BHOH617
AGLY16
AGLY17
AHOH1242
BARG14
BGLY16
BGLY17
BHOH515
BHOH525

site_idAC2
残基数3
詳細BINDING SITE FOR RESIDUE PO4 A 502
鎖名残基
ALYS7
AARG8
AHOH1225

site_idAC3
残基数7
詳細BINDING SITE FOR RESIDUE PO4 B 503
鎖名残基
AGLY68
AHIS69
ALYS70
AHOH1210
AHOH1249
BPRO1
BLYS55

site_idAC4
残基数5
詳細BINDING SITE FOR RESIDUE PO4 A 504
鎖名残基
AMET36
AASN37
BPRO39
BGLY40
BHOH621

site_idAC5
残基数6
詳細BINDING SITE FOR RESIDUE PO4 A 505
鎖名残基
ALYS20
AGLU21
AASN83
AHOH1219
AHOH1226
BHOH616

site_idAC6
残基数19
詳細BINDING SITE FOR RESIDUE 017 A 1200
鎖名残基
AASP25
AGLY27
AALA28
AASP29
AASP30
AGLY48
AGLY49
AILE50
AHOH1203
AHOH1311
BASP25
BGLY27
BALA28
BASP30
BVAL32
BGLY48
BGLY49
BVAL82
BILE84

UniProtにおけるモチーフ・データベースPROSITEからの機能情報
site_idPS00141
残基数12
詳細ASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. ALLDTGADDTVL
鎖名残基詳細
AALA22-LEU33

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数2
詳細SITE: Cleavage; by viral protease => ECO:0000250
鎖名残基詳細
AGLY78
BGLY78

site_idSWS_FT_FI2
残基数2
詳細MOD_RES: Phosphotyrosine; by host => ECO:0000250
鎖名残基詳細
AGLY78
BGLY78

CSAにおける酵素触媒機能の情報
site_idCSA1
残基数4
詳細Annotated By Reference To The Literature 1a30
鎖名残基詳細
AASP25
ATHR26
BASP25
BTHR26

site_idCSA2
残基数2
詳細Annotated By Reference To The Literature 1a30
鎖名残基詳細
AASP25
BASP25

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件を2024-09-18に公開中

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