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1INY

A SIALIC ACID DERIVED PHOSPHONATE ANALOG INHIBITS DIFFERENT STRAINS OF INFLUENZA VIRUS NEURAMINIDASE WITH DIFFERENT EFFICIENCIES

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004308molecular_functionexo-alpha-sialidase activity
A0005975biological_processcarbohydrate metabolic process
A0016020cellular_componentmembrane
A0033644cellular_componenthost cell membrane
A0046761biological_processviral budding from plasma membrane
A0055036cellular_componentvirion membrane
PDBデータベースに由来する情報
site_idCAT
残基数11
詳細SUBSTRATE (SIALIC ACID) BINDING RESIDUES IN CATALYTIC SITE
鎖名残基
AARG118
AARG371
ATYR405
AGLU119
AASP151
AARG152
ATRP179
AILE223
AARG225
AGLU277
AARG293

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数1
詳細ACT_SITE: Proton donor/acceptor => ECO:0000255|HAMAP-Rule:MF_04071
鎖名残基詳細
AASP151

site_idSWS_FT_FI2
残基数1
詳細ACT_SITE: Nucleophile => ECO:0000255|HAMAP-Rule:MF_04071
鎖名残基詳細
ATYR405

site_idSWS_FT_FI3
残基数5
詳細BINDING: BINDING => ECO:0000255|HAMAP-Rule:MF_04071
鎖名残基詳細
AARG118
AARG152
AGLU277
AARG293
AARG371

site_idSWS_FT_FI4
残基数4
詳細BINDING: BINDING => ECO:0000255|HAMAP-Rule:MF_04071, ECO:0000269|PubMed:23429702, ECO:0000269|PubMed:7549872, ECO:0000269|PubMed:8371267, ECO:0000269|PubMed:9342319
鎖名残基詳細
AASP294
AGLY298
AASP325
AASN347

site_idSWS_FT_FI5
残基数3
詳細CARBOHYD: N-linked (GlcNAc...) asparagine; by host => ECO:0000255|HAMAP-Rule:MF_04071, ECO:0000269|PubMed:23429702, ECO:0000269|PubMed:7549872, ECO:0000269|PubMed:9342319
鎖名残基詳細
AASN86
AASN146
AASN201

CSAにおける酵素触媒機能の情報
site_idCSA1
残基数2
詳細Annotated By Reference To The Literature 1a4g
鎖名残基詳細
AGLU278
AASP151

site_idMCSA1
残基数5
詳細M-CSA 828
鎖名残基詳細
AASP151activator, electrostatic stabiliser, increase acidity, increase nucleophilicity, proton acceptor, proton donor
AGLU278activator, electrostatic stabiliser, increase nucleophilicity, promote heterolysis, proton acceptor, proton donor
AARG293electrostatic stabiliser
AARG371electrostatic stabiliser
ATYR405electrostatic stabiliser, nucleofuge, nucleophile, proton acceptor, proton donor

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件を2024-09-18に公開中

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