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5Q06

Human liver fructose-1,6-bisphosphatase 1 (fructose 1,6-bisphosphate 1-phosphatase, E.C.3.1.3.11) complexed with the allosteric inhibitor 1-(5-bromo-1,3-thiazol-2-yl)-3-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]sulfonylurea

Experimental procedure
実験手法SINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsSLS BEAMLINE X10SA
Synchrotron siteSLS
BeamlineX10SA
Temperature [K]100
Detector technologyCCD
Collection date2006-03-17
DetectorMAR CCD 165 mm
Wavelength(s)0.987
Spacegroup nameP 21 21 21
格子定数 [Å]67.506, 83.695, 278.843
格子定数 [度]90.00, 90.00, 90.00
精密化法
残基19.986 - 2.400
R因子0.1713
Rwork0.168
R-free0.23380
Structure solution methodMOLECULAR REPLACEMENT
結合長の平均二乗偏差(RMSD) [Å]0.008
結合角の平均二乗偏差(RMSD) [度]0.998
Refinement softwarePHENIX (1.11.1_2575)
Quality characteristics
 Overall
分解能 [Å] (低)19.986
分解能 [Å] (高)2.400
独立反射数62733
完全性 [%]100.0
結晶化条件
結晶ID方法pH温度溶液条件
1VAPOR DIFFUSION, SITTING DROP73000.1M HEPES pH 7.0, 0.1M AMMONIUM ACETATE, 12% PEG 3350

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件を2024-09-18に公開中

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