7LVK
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![BU of 7lvk by Molmil](/molmil-images/mine/7lvk) | Cfr-modified 50S subunit from Escherichia coli | Descriptor: | 23S rRNA, 50S ribosomal protein L13, 50S ribosomal protein L14, ... | Authors: | Stojkovic, V, Myasnikov, A.G, Frost, A, Fujimori, D.G. | Deposit date: | 2021-02-25 | Release date: | 2021-12-15 | Last modified: | 2023-11-15 | Method: | ELECTRON MICROSCOPY (2.2 Å) | Cite: | Investigating antibiotic resistance of a ribosomal-RNA methylating enzyme through directed evolution To Be Published
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7M1A
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![BU of 7m1a by Molmil](/molmil-images/mine/7m1a) | SusE-like protein BT2857 | Descriptor: | 1,2-ETHANEDIOL, CALCIUM ION, Galactose-binding like protein | Authors: | Suits, M.D.L. | Deposit date: | 2021-03-12 | Release date: | 2021-04-21 | Last modified: | 2021-07-28 | Method: | X-RAY DIFFRACTION (1.42 Å) | Cite: | Analysis of Two SusE-Like Enzymes From Bacteroides thetaiotaomicron Reveals a Potential Degradative Capacity for This Protein Family. Front Microbiol, 12, 2021
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7M1B
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![BU of 7m1b by Molmil](/molmil-images/mine/7m1b) | SusE-like protein BT2857 | Descriptor: | 1,2-ETHANEDIOL, Galactose-binding-like protein | Authors: | Suits, M.D.L. | Deposit date: | 2021-03-12 | Release date: | 2021-04-21 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (1.5 Å) | Cite: | Analysis of Two SusE-Like Enzymes From Bacteroides thetaiotaomicron Reveals a Potential Degradative Capacity for This Protein Family. Front Microbiol, 12, 2021
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7M2T
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![BU of 7m2t by Molmil](/molmil-images/mine/7m2t) | |
7M2V
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![BU of 7m2v by Molmil](/molmil-images/mine/7m2v) | |
7M3L
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![BU of 7m3l by Molmil](/molmil-images/mine/7m3l) | |
7M3R
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![BU of 7m3r by Molmil](/molmil-images/mine/7m3r) | |
7M3T
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![BU of 7m3t by Molmil](/molmil-images/mine/7m3t) | |
7M4W
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![BU of 7m4w by Molmil](/molmil-images/mine/7m4w) | A. baumannii Ribosome-Eravacycline complex: Empty 70S | Descriptor: | 16s Ribosomal RNA, 23s ribosomal RNA, 30S ribosomal protein S10, ... | Authors: | Morgan, C.E, Yu, E.W. | Deposit date: | 2021-03-22 | Release date: | 2021-05-19 | Last modified: | 2024-03-06 | Method: | ELECTRON MICROSCOPY (2.55 Å) | Cite: | Cryo-EM Determination of Eravacycline-Bound Structures of the Ribosome and the Multidrug Efflux Pump AdeJ of Acinetobacter baumannii. Mbio, 12, 2021
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7M4X
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![BU of 7m4x by Molmil](/molmil-images/mine/7m4x) | A. baumannii Ribosome-Eravacycline complex: P-site tRNA 70S | Descriptor: | 16s Ribosomal RNA, 23s ribosomal RNA, 30S ribosomal protein S10, ... | Authors: | Morgan, C.E, Yu, E.W. | Deposit date: | 2021-03-22 | Release date: | 2021-05-19 | Last modified: | 2024-03-06 | Method: | ELECTRON MICROSCOPY (2.66 Å) | Cite: | Cryo-EM Determination of Eravacycline-Bound Structures of the Ribosome and the Multidrug Efflux Pump AdeJ of Acinetobacter baumannii. Mbio, 12, 2021
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7M4Y
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![BU of 7m4y by Molmil](/molmil-images/mine/7m4y) | A. baumannii Ribosome-Eravacycline complex: E-site tRNA 70S | Descriptor: | 16s Ribosomal RNA, 23s ribosomal RNA, 30S ribosomal protein S10, ... | Authors: | Morgan, C.E, Yu, E.W. | Deposit date: | 2021-03-22 | Release date: | 2021-05-19 | Last modified: | 2024-03-06 | Method: | ELECTRON MICROSCOPY (2.5 Å) | Cite: | Cryo-EM Determination of Eravacycline-Bound Structures of the Ribosome and the Multidrug Efflux Pump AdeJ of Acinetobacter baumannii. Mbio, 12, 2021
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7M4Z
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![BU of 7m4z by Molmil](/molmil-images/mine/7m4z) | A. baumannii Ribosome-Eravacycline complex: hpf-bound 70S | Descriptor: | 16s Ribosomal RNA, 23s ribosomal RNA, 30S ribosomal protein S10, ... | Authors: | Morgan, C.E, Yu, E.W. | Deposit date: | 2021-03-22 | Release date: | 2021-05-19 | Last modified: | 2024-03-06 | Method: | ELECTRON MICROSCOPY (2.92 Å) | Cite: | Cryo-EM Determination of Eravacycline-Bound Structures of the Ribosome and the Multidrug Efflux Pump AdeJ of Acinetobacter baumannii. Mbio, 12, 2021
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7M50
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![BU of 7m50 by Molmil](/molmil-images/mine/7m50) | |
7M54
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![BU of 7m54 by Molmil](/molmil-images/mine/7m54) | |
7M57
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![BU of 7m57 by Molmil](/molmil-images/mine/7m57) | |
7M5D
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![BU of 7m5d by Molmil](/molmil-images/mine/7m5d) | |
7M6A
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![BU of 7m6a by Molmil](/molmil-images/mine/7m6a) | High resolution structure of the membrane embedded skeletal muscle ryanodine receptor | Descriptor: | ADENOSINE-5'-TRIPHOSPHATE, CAFFEINE, CALCIUM ION, ... | Authors: | Melville, Z, Kim, K, Clarke, O.B, Marks, A.R. | Deposit date: | 2021-03-25 | Release date: | 2021-09-08 | Last modified: | 2022-01-19 | Method: | ELECTRON MICROSCOPY (3.36 Å) | Cite: | High-resolution structure of the membrane-embedded skeletal muscle ryanodine receptor. Structure, 30, 2022
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7M6L
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![BU of 7m6l by Molmil](/molmil-images/mine/7m6l) | High resolution structure of the membrane embedded skeletal muscle ryanodine receptor | Descriptor: | ADENOSINE-5'-TRIPHOSPHATE, CAFFEINE, CALCIUM ION, ... | Authors: | Melville, Z, Kim, K, Clarke, O.B, Marks, A.R. | Deposit date: | 2021-03-25 | Release date: | 2021-08-18 | Last modified: | 2022-01-19 | Method: | ELECTRON MICROSCOPY (3.98 Å) | Cite: | High-resolution structure of the membrane-embedded skeletal muscle ryanodine receptor. Structure, 30, 2022
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7MD2
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![BU of 7md2 by Molmil](/molmil-images/mine/7md2) | The F1 region of ammocidin-bound Saccharomyces cerevisiae ATP synthase | Descriptor: | (3~{E},5~{Z},7~{E},9~{R},10~{S},11~{E},13~{E},15~{E},17~{R},18~{S},20~{S})-20-[(1~{R})-1-[(2~{S},3~{R},4~{R},5~{S},6~{R})-5-[(2~{S},4~{S},5~{S},6~{R})-5-[(2~{S},4~{R},5~{R},6~{R})-4,6-dimethyl-4,5-bis(oxidanyl)oxan-2-yl]oxy-6-methyl-4-oxidanyl-oxan-2-yl]oxy-3-methoxy-6-(3-methoxypropyl)-5-methyl-2,4-bis(oxidanyl)oxan-2-yl]ethyl]-5,18-dimethoxy-3,7,9,11,13,15-hexamethyl-10-[(2~{R},3~{S},4~{R},5~{R},6~{S})-6-methyl-3,4,5-tris(oxidanyl)oxan-2-yl]oxy-17-oxidanyl-1-oxacycloicosa-3,5,7,11,13,15-hexaen-2-one, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase subunit alpha, ... | Authors: | Guo, H, Rubinstein, J.L. | Deposit date: | 2021-04-03 | Release date: | 2021-08-11 | Last modified: | 2024-05-29 | Method: | ELECTRON MICROSCOPY (3.1 Å) | Cite: | A Family of Glycosylated Macrolides Selectively Target Energetic Vulnerabilities in Leukemia Biorxiv, 2021
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7MD3
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![BU of 7md3 by Molmil](/molmil-images/mine/7md3) | The F1 region of apoptolidin-bound Saccharomyces cerevisiae ATP synthase | Descriptor: | (3~{E},5~{E},7~{E},9~{R},10~{R},11~{E},13~{E},17~{S},18~{S},20~{S})-18-methoxy-20-[(~{R})-[(2~{R},3~{R},4~{S},5~{R},6~{R})-6-[(2~{R})-3-methoxy-2-[(2~{R},4~{S},5~{S},6~{S})-5-[(2~{S},4~{R},5~{R},6~{R})-4-methoxy-6-methyl-5-oxidanyl-oxan-2-yl]oxy-4,6-dimethyl-4-oxidanyl-oxan-2-yl]oxy-propyl]-3,5-dimethyl-2,4-bis(oxidanyl)oxan-2-yl]-oxidanyl-methyl]-10-[(2~{R},3~{S},4~{S},5~{R},6~{S})-5-methoxy-6-methyl-3,4-bis(oxidanyl)oxan-2-yl]oxy-3,5,7,9,13-pentamethyl-17-oxidanyl-1-oxacycloicosa-3,5,7,11,13-pentaen-2-one, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase subunit alpha, ... | Authors: | Guo, H, Rubinstein, J.L. | Deposit date: | 2021-04-03 | Release date: | 2021-08-11 | Last modified: | 2024-05-29 | Method: | ELECTRON MICROSCOPY (3.3 Å) | Cite: | A Family of Glycosylated Macrolides Selectively Target Energetic Vulnerabilities in Leukemia Biorxiv, 2021
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7MD7
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![BU of 7md7 by Molmil](/molmil-images/mine/7md7) | Crystal structure of the Thermus thermophilus 70S ribosome in complex with triphenylphosphonium analog of chloramphenicol CAM-C4-TPP and protein Y (YfiA) at 2.80A resolution | Descriptor: | (4S)-2-METHYL-2,4-PENTANEDIOL, 16S Ribosomal RNA, 23S Ribosomal RNA, ... | Authors: | Chen, C.-W, Pavlova, J.A, Lukianov, D.A, Tereshchenkov, A.G, Makarov, G.I, Khairullina, Z.Z, Tashlitsky, V.N, Paleskava, A, Konevega, A.L, Bogdanov, A.A, Osterman, I.A, Sumbatyan, N.V, Polikanov, Y.S. | Deposit date: | 2021-04-03 | Release date: | 2021-04-21 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Binding and Action of Triphenylphosphonium Analog of Chloramphenicol upon the Bacterial Ribosome. Antibiotics, 10, 2021
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7MDZ
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![BU of 7mdz by Molmil](/molmil-images/mine/7mdz) | 80S rabbit ribosome stalled with benzamide-CHX | Descriptor: | 18S rRNA, 28S rRNA, 40S ribosomal protein S21, ... | Authors: | Koga, Y, Hoang, E.M, Park, Y, Keszei, A.F.A, Murray, J, Shao, S, Liau, B.B. | Deposit date: | 2021-04-06 | Release date: | 2021-09-01 | Last modified: | 2021-09-15 | Method: | ELECTRON MICROSCOPY (3.2 Å) | Cite: | Discovery of C13-Aminobenzoyl Cycloheximide Derivatives that Potently Inhibit Translation Elongation. J.Am.Chem.Soc., 143, 2021
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7MF0
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![BU of 7mf0 by Molmil](/molmil-images/mine/7mf0) | Co-crystal structure of PERK with inhibitor (R)-2-amino-N-cyclopropyl-5-(4-(2-(3,5-difluorophenyl)-2-hydroxyacetamido)-2-methylphenyl)nicotinamide | Descriptor: | 2-amino-N-cyclopropyl-5-(4-{[(2R)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamide, Eukaryotic translation initiation factor 2-alpha kinase 3,Eukaryotic translation initiation factor 2-alpha kinase 3 | Authors: | Wiens, B, Koszelak-Rosenblum, M, Surman, M.D, Zhu, G, Mulvihill, M.J. | Deposit date: | 2021-04-08 | Release date: | 2021-05-19 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.809 Å) | Cite: | Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors. Bioorg.Med.Chem.Lett., 43, 2021
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7MFJ
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![BU of 7mfj by Molmil](/molmil-images/mine/7mfj) | Structural Characterization of Beta Cyanoalanine Synthase from Tetranychus Urticae | Descriptor: | ACETATE ION, Beta-cyanoalanine synthase, PYRIDOXAL-5'-PHOSPHATE | Authors: | Daneshian, L, Schlachter, C, Dermauw, W, Wybouw, N, Van Leeuwen, T, Chruszcz, M. | Deposit date: | 2021-04-09 | Release date: | 2021-11-24 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.351 Å) | Cite: | Structural and functional characterization of beta-cyanoalanine synthase from Tetranychus urticae. Insect Biochem.Mol.Biol., 142, 2022
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7MFM
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![BU of 7mfm by Molmil](/molmil-images/mine/7mfm) | Glutamate synthase, glutamate dehydrogenase counter-enzyme complex | Descriptor: | FE3-S4 CLUSTER, FLAVIN MONONUCLEOTIDE, FLAVIN-ADENINE DINUCLEOTIDE, ... | Authors: | Jayaraman, V, Lee, D.J, Elad, N, Fraser, J.S, Tawfik, D.S. | Deposit date: | 2021-04-10 | Release date: | 2022-01-05 | Last modified: | 2022-02-16 | Method: | ELECTRON MICROSCOPY (2.42 Å) | Cite: | A counter-enzyme complex regulates glutamate metabolism in Bacillus subtilis. Nat.Chem.Biol., 18, 2022
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