Entry Database : PDB / ID : 4bqh Structure visualization Downloads & linksTitle Crystal structure of the uridine diphosphate N-acetylglucosamine pyrophosphorylase from Trypanosoma brucei in complex with inhibitor ComponentsUDP-N-ACETYLGLUCOSAMINE PYROPHOSPHORYLASE Details Keywords TRANSFERASE / INHIBITORFunction / homology Function and homology informationFunction Domain/homology Component
nucleotide-sugar biosynthetic process / UDP-N-acetylglucosamine diphosphorylase / UDP-N-acetylglucosamine diphosphorylase activity / UDP-glucose metabolic process / UDP-N-acetylglucosamine biosynthetic process / glycosome / nucleotidyltransferase activity / cytoplasm Similarity search - Function UDP-sugar pyrophosphorylase / UDPGP family / UTP--glucose-1-phosphate uridylyltransferase / Spore Coat Polysaccharide Biosynthesis Protein SpsA; Chain A / Spore Coat Polysaccharide Biosynthesis Protein SpsA; Chain A / Nucleotide-diphospho-sugar transferases / Alpha-Beta Complex / Alpha Beta Similarity search - Domain/homologyBiological species TRYPANOSOMA BRUCEI (eukaryote)Method X-RAY DIFFRACTION / SYNCHROTRON / MOLECULAR REPLACEMENT / Resolution : 1.75 Å DetailsAuthors Fang, W. / Raimi, O.G. / vanAalten, D.M.F. CitationJournal : Acs Chem.Biol. / Year : 2013Title : A Novel Allosteric Inhibitor of the Uridine Diphosphate N-Acetylglucosamine Pyrophosphorylase from Trypanosoma Brucei.Authors : Urbaniak, M.D. / Collie, I.T. / Fang, W. / Aristotelous, T. / Eskilsson, S. / Raimi, O.G. / Harrison, J. / Hopkins Navratolova, I. / Frearson, J.A. / Van Aalten, D.M.F. / Ferguson, M.A.J. History Deposition May 30, 2013 Deposition site : PDBE / Processing site : PDBERevision 1.0 Jul 17, 2013 Provider : repository / Type : Initial releaseRevision 1.1 Oct 9, 2013 Group : Database referencesRevision 1.2 Dec 20, 2023 Group : Data collection / Database references ... Data collection / Database references / Derived calculations / Other / Refinement description Category : chem_comp_atom / chem_comp_bond ... chem_comp_atom / chem_comp_bond / database_2 / pdbx_database_status / pdbx_initial_refinement_model / struct_site Item : _database_2.pdbx_DOI / _database_2.pdbx_database_accession ... _database_2.pdbx_DOI / _database_2.pdbx_database_accession / _pdbx_database_status.status_code_sf / _struct_site.pdbx_auth_asym_id / _struct_site.pdbx_auth_comp_id / _struct_site.pdbx_auth_seq_id
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