登録情報 | データベース: PDB / ID: 6yqs |
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タイトル | BRD9 with methylpiperazinyl-benzyl-amino-dimethylpyridazinone |
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要素 | Bromodomain-containing protein 9 |
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キーワード | TRANSCRIPTION / BRD9 / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN |
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機能・相同性 | 機能・相同性情報
GBAF complex / SWI/SNF complex / positive regulation of stem cell population maintenance / negative regulation of cell differentiation / lysine-acetylated histone binding / nucleic acid binding / chromatin remodeling / positive regulation of cell population proliferation / chromatin / regulation of transcription by RNA polymerase II ...GBAF complex / SWI/SNF complex / positive regulation of stem cell population maintenance / negative regulation of cell differentiation / lysine-acetylated histone binding / nucleic acid binding / chromatin remodeling / positive regulation of cell population proliferation / chromatin / regulation of transcription by RNA polymerase II / nucleoplasm / nucleus類似検索 - 分子機能 Protein of unknown function DUF3512 / Domain of unknown function (DUF3512) / : / Bromodomain / Bromodomain profile. / bromo domain / Bromodomain / Bromodomain-like superfamily類似検索 - ドメイン・相同性 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / フーリエ合成 / 解像度: 1.683 Å |
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データ登録者 | Chung, C. |
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引用 | ジャーナル: J.Med.Chem. / 年: 2020 タイトル: Application of Atypical Acetyl-lysine Methyl Mimetics in the Development of Selective Inhibitors of the Bromodomain-Containing Protein 7 (BRD7)/Bromodomain-Containing Protein 9 (BRD9) Bromodomains. 著者: Clegg, M.A. / Bamborough, P. / Chung, C.W. / Craggs, P.D. / Gordon, L. / Grandi, P. / Leveridge, M. / Lindon, M. / Liwicki, G.M. / Michon, A.M. / Molnar, J. / Rioja, I. / Soden, P.E. / ...著者: Clegg, M.A. / Bamborough, P. / Chung, C.W. / Craggs, P.D. / Gordon, L. / Grandi, P. / Leveridge, M. / Lindon, M. / Liwicki, G.M. / Michon, A.M. / Molnar, J. / Rioja, I. / Soden, P.E. / Theodoulou, N.H. / Werner, T. / Tomkinson, N.C.O. / Prinjha, R.K. / Humphreys, P.G. |
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履歴 | 登録 | 2020年4月18日 | 登録サイト: PDBE / 処理サイト: PDBE |
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改定 1.0 | 2021年3月24日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2024年5月15日 | Group: Data collection / Database references / Derived calculations カテゴリ: atom_type / chem_comp_atom ...atom_type / chem_comp_atom / chem_comp_bond / database_2 Item: _atom_type.pdbx_N_electrons / _atom_type.pdbx_scat_Z ..._atom_type.pdbx_N_electrons / _atom_type.pdbx_scat_Z / _database_2.pdbx_DOI / _database_2.pdbx_database_accession |
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