- PDB-6ekn: Crystal structure of MMP12 in complex with inhibitor BE7. -
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IDまたはキーワード:
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基本情報
登録情報
データベース: PDB / ID: 6ekn
タイトル
Crystal structure of MMP12 in complex with inhibitor BE7.
要素
Macrophage metalloelastase
キーワード
HYDROLASE / metzincin / carboxylate inhibitor alternative zinc-binding groups
機能・相同性
機能・相同性情報
macrophage elastase / negative regulation of endothelial cell-matrix adhesion via fibronectin / bronchiole development / positive regulation of epithelial cell proliferation involved in wound healing / elastin catabolic process / regulation of defense response to virus by host / positive regulation of type I interferon-mediated signaling pathway / wound healing, spreading of epidermal cells / lung alveolus development / negative regulation of type I interferon-mediated signaling pathway ...macrophage elastase / negative regulation of endothelial cell-matrix adhesion via fibronectin / bronchiole development / positive regulation of epithelial cell proliferation involved in wound healing / elastin catabolic process / regulation of defense response to virus by host / positive regulation of type I interferon-mediated signaling pathway / wound healing, spreading of epidermal cells / lung alveolus development / negative regulation of type I interferon-mediated signaling pathway / positive regulation of interferon-alpha production / response to amyloid-beta / Collagen degradation / collagen catabolic process / extracellular matrix disassembly / core promoter sequence-specific DNA binding / collagen binding / Degradation of the extracellular matrix / extracellular matrix / extracellular matrix organization / cellular response to virus / metalloendopeptidase activity / protein import into nucleus / endopeptidase activity / sequence-specific DNA binding / serine-type endopeptidase activity / calcium ion binding / negative regulation of transcription by RNA polymerase II / positive regulation of transcription by RNA polymerase II / proteolysis / extracellular space / zinc ion binding / extracellular region / nucleus / cytoplasm 類似検索 - 分子機能
解像度: 1.2→36.74 Å / Cor.coef. Fo:Fc: 0.985 / Cor.coef. Fo:Fc free: 0.979 / SU B: 1.786 / SU ML: 0.031 / 交差検証法: THROUGHOUT / σ(F): 0 / ESU R: 0.04 / ESU R Free: 0.04 / 詳細: HYDROGENS HAVE BEEN ADDED IN THE RIDING POSITIONS