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-Structure paper
Title | Structural Analysis and Development of Notum Fragment Screening Hits. |
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Journal, issue, pages | Acs Chem Neurosci, Vol. 13, Page 2060-2077, Year 2022 |
Publish date | Dec 2, 2020 (structure data deposition date) |
![]() | Zhao, Y. / Mahy, W. / Willis, N.J. / Woodward, H.L. / Steadman, D. / Bayle, E.D. / Atkinson, B.N. / Sipthorp, J. / Vecchia, L. / Ruza, R.R. ...Zhao, Y. / Mahy, W. / Willis, N.J. / Woodward, H.L. / Steadman, D. / Bayle, E.D. / Atkinson, B.N. / Sipthorp, J. / Vecchia, L. / Ruza, R.R. / Harlos, K. / Jeganathan, F. / Constantinou, S. / Costa, A. / Kjaer, S. / Bictash, M. / Salinas, P.C. / Whiting, P. / Vincent, J.P. / Fish, P.V. / Jones, E.Y. |
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Methods | X-ray diffraction |
Resolution | 1.24 - 1.94 Å |
Structure data | ![]() PDB-7b4x: ![]() PDB-7b84: ![]() PDB-7b86: ![]() PDB-7b87: ![]() PDB-7b89: ![]() PDB-7b8c: ![]() PDB-7b8d: ![]() PDB-7b8f: ![]() PDB-7b8g: ![]() PDB-7b8j: ![]() PDB-7b8k: ![]() PDB-7b8l: ![]() PDB-7b8m: ![]() PDB-7b8n: ![]() PDB-7b8o: ![]() PDB-7b8u: ![]() PDB-7b8x: ![]() PDB-7b8y: ![]() PDB-7b8z: ![]() PDB-7b98: ![]() PDB-7b99: ![]() PDB-7b9d: ![]() PDB-7b9i: ![]() PDB-7b9n: ![]() PDB-7b9u: ![]() PDB-7ba1: ![]() PDB-7bac: ![]() PDB-7bap: ![]() PDB-7bc8: ![]() PDB-7bc9: ![]() PDB-7bcc: ![]() PDB-7bcd: ![]() PDB-7bcf: ![]() PDB-7bch: ![]() PDB-7bci: ![]() PDB-7bck: ![]() PDB-7bcl: ![]() PDB-7bd2: ![]() PDB-7bd3: ![]() PDB-7bd4: ![]() PDB-7bd5: ![]() PDB-7bd6: ![]() PDB-7bd8: ![]() PDB-7bd9: ![]() PDB-7bda: ![]() PDB-7bdb: ![]() PDB-7bdc: ![]() PDB-7bdd: ![]() PDB-7bdf: ![]() PDB-7bdg: ![]() PDB-7bdh: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-DMS: ![]() ChemComp-EDO: ![]() ChemComp-SWT: ![]() ChemComp-HOH: ![]() ChemComp-NAG: ![]() ChemComp-JFS: ![]() ChemComp-AW7: ![]() ChemComp-JFV: ![]() ChemComp-T1Z: ![]() ChemComp-GRV: ![]() ChemComp-SFY: ![]() ChemComp-RYM: ![]() ChemComp-MJW: ![]() ChemComp-BP4: ![]() ChemComp-AXV: ![]() ChemComp-AY4: ![]() ChemComp-GQM: ![]() ChemComp-GOL: ![]() ChemComp-T2E: ![]() ChemComp-T1W: ![]() ChemComp-RUY: ![]() ChemComp-U3K: ![]() ChemComp-T2H: ![]() ChemComp-A6Z: ![]() ChemComp-EJW: ![]() ChemComp-B1A: ![]() ChemComp-T3N: ![]() ChemComp-T3T: ![]() ChemComp-N9J: ![]() ChemComp-O3D: ![]() ChemComp-S1V: ![]() ChemComp-LO5: ![]() ChemComp-S4V: ![]() ChemComp-TAH: ![]() ChemComp-UR4: ![]() ChemComp-TB5: ![]() ChemComp-T9Z: ![]() ChemComp-T9W: ![]() ChemComp-T9Q: ![]() ChemComp-GVV: ![]() ChemComp-T9B: ![]() ChemComp-T9K: ![]() ChemComp-NUM: ![]() ChemComp-TE5: ![]() ChemComp-JHJ: ![]() ChemComp-YI6: ![]() ChemComp-JH7: ![]() ChemComp-QL5: ![]() ChemComp-GW1: ![]() ChemComp-O1J: ![]() ChemComp-NW7: ![]() ChemComp-WNA: ![]() ChemComp-TE8: ![]() ChemComp-TEH: ![]() ChemComp-TEK: ![]() ChemComp-TEZ: |
Source |
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![]() | HYDROLASE / Notum Inhibitor complex / Notum Fragment / Notum Inhibitor / Notum Inhibitor Wnt / Notum Inhibitor Fragment Screen |