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| Title | Structure-guided development of a potent human B0AT1 inhibitor effective in a mouse model of phenylketonuria |
|---|---|
| Journal, issue, pages | To Be Published |
| Publish date | Dec 7, 2024 (structure data deposition date) |
Authors | Imazu T / Akashi T / Hiraizumi M / Inui Y / Sasaki W / Takahashi T / Todoroki H / Kumanomidou T / Hisano H / Asada H ...Imazu T / Akashi T / Hiraizumi M / Inui Y / Sasaki W / Takahashi T / Todoroki H / Kumanomidou T / Hisano H / Asada H / Kusakizako T / Nishizawa T / Iwata S / Nureki O / Miyaguchi I |
External links | Search PubMed |
| Methods | EM (single particle) |
| Resolution | 2.66 - 2.87 Å |
| Structure data | EMDB-62627, PDB-9kxt: EMDB-62628, PDB-9kxu: EMDB-62629, PDB-9kxv: EMDB-62630, PDB-9kxw: EMDB-62631, PDB-9kxx: EMDB-62632, PDB-9kxy: |
| Chemicals | ![]() PDB-1l6u: ![]() ChemComp-NAG: ![]() ChemComp-HOH: ![]() PDB-1l6v: ![]() PDB-1l6w: ![]() ChemComp-NA: |
| Source |
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Keywords | TRANSPORT PROTEIN / Inhibitor / amino acid transporter / SLC6 |
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homo sapiens (human)
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