Systematic Design of Adenosine Analogs as Inhibitors of a Clostridioides difficile- Specific DNA Adenine Methyltransferase Required for Normal Sporulation and Persistence.
PDB-8cxs: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor MTA 手法: X-RAY DIFFRACTION / 解像度: 2.49 Å
PDB-8cxt: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor N6-benzyladenosine (Compound 1) 手法: X-RAY DIFFRACTION / 解像度: 2.61 Å
PDB-8cxu: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 2 手法: X-RAY DIFFRACTION / 解像度: 2.28 Å
PDB-8cxv: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 3 手法: X-RAY DIFFRACTION / 解像度: 2.26 Å
PDB-8cxw: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor piclidenoson (Compound 4) 手法: X-RAY DIFFRACTION / 解像度: 2.78 Å
PDB-8cxx: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 6 手法: X-RAY DIFFRACTION / 解像度: 2.34 Å
PDB-8cxy: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor N6-(2-Phenethyl)adenosine (Compound 8) 手法: X-RAY DIFFRACTION / 解像度: 2.19 Å
PDB-8cxz: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor N6-(3-Phenylpropyl)adenosine (Compound 14) 手法: X-RAY DIFFRACTION / 解像度: 2.35 Å
PDB-8cy0: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor MC4756 (Compound 178) 手法: X-RAY DIFFRACTION / 解像度: 2.65 Å
PDB-8cy1: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 19 手法: X-RAY DIFFRACTION / 解像度: 2.38 Å
PDB-8cy2: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor APNEA (Compound 9) 手法: X-RAY DIFFRACTION / 解像度: 2.81 Å
PDB-8cy3: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 15 手法: X-RAY DIFFRACTION / 解像度: 2.65 Å
PDB-8cy4: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 16 手法: X-RAY DIFFRACTION / 解像度: 2.34 Å
PDB-8cy5: CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Compound 39 手法: X-RAY DIFFRACTION / 解像度: 2.5 Å