タイトル | X-ray structures of AMPA receptor-cone snail toxin complexes illuminate activation mechanism. |
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ジャーナル・号・ページ | Science, Vol. 345, Page 1021-1026, Year 2014 |
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掲載日 | 2014年7月25日 (構造データの登録日) |
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著者 | Chen, L. / Durr, K.L. / Gouaux, E. |
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リンク | Science / PubMed:25103405 |
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手法 | X線回折 |
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解像度 | 1.58 - 3.7 Å |
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構造データ | PDB-4u5b: Crystal structure of GluA2 A622T, con-ikot-ikot snail toxin, partial agonist KA and postitive modulator (R,R)-2b complex 手法: X-RAY DIFFRACTION / 解像度: 3.5037 Å PDB-4u5c: Crystal structure of GluA2, con-ikot-ikot snail toxin, partial agonist FW and postitive modulator (R,R)-2b complex 手法: X-RAY DIFFRACTION / 解像度: 3.6883 Å PDB-4u5d: Crystal structure of GluA2, con-ikot-ikot snail toxin, partial agonist KA and postitive modulator (R,R)-2b complex 手法: X-RAY DIFFRACTION / 解像度: 3.5757 Å PDB-4u5e: Crystal structure of GluA2 T625G, con-ikot-ikot snail toxin, partial agonist KA and postitive modulator (R,R)-2b complex 手法: X-RAY DIFFRACTION / 解像度: 3.5073 Å PDB-4u5f: Crystal structure of GluA2, con-ikot-ikot snail toxin, partial agonist KA and postitive modulator (R,R)-2b complex, GluA2cryst2 construct 手法: X-RAY DIFFRACTION / 解像度: 3.7 Å PDB-4u5g: Crystal structure of con-ikot-ikot toxin 手法: X-RAY DIFFRACTION / 解像度: 2.1997 Å PDB-4u5h: crystal structure of con-ikot-ikot toxin 手法: X-RAY DIFFRACTION / 解像度: 1.58 Å |
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化合物 | ChemComp-KAI: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE / カイニン酸 / 神経伝達物質, アゴニスト*YM
ChemComp-FWF: N,N'-[biphenyl-4,4'-diyldi(2R)propane-2,1-diyl]dipropane-2-sulfonamide
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由来 | - rattus norvegicus (ドブネズミ)
- conus striatus (ニシキミナシ)
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キーワード | Transport protein/toxin / AMPA receptor / Transport protein-toxin complex / AMPA receptors / TOXIN |
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