タイトル | Novel Blocker of Onco SK3 Channels Derived from Scorpion Toxin Tamapin and Active against Migration of Cancer Cells |
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ジャーナル・号・ページ | Acs Med. Chem. Lett., Year 2020 |
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掲載日 | 2018年4月16日 (構造データの登録日) |
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著者 | Mayorga-Flores, M. / Chantome, A. / Melchor Meneses, C.M. / Domingo, I. / Titaux Delgado, G. / Galindo Murillo, R. / Vandier, C. / del Rio Portilla, F. |
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リンク | Acs Med. Chem. Lett. / PubMedで検索 |
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手法 | NMR (溶液) |
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構造データ | PDB-6d3t: NMR solution structure of tamapin, mutant DP30 手法: SOLUTION NMR PDB-6d8h: NMR solution structure of tamapin, mutant Y31+N 手法: SOLUTION NMR PDB-6d8q: NMR solution structure of tamapin, mutant DP30/Y31+N 手法: SOLUTION NMR PDB-6d8r: NMR solution structure of tamapin, mutant E25K 手法: SOLUTION NMR PDB-6d8s: NMR solution structure of tamapin, mutant K27E 手法: SOLUTION NMR PDB-6d8t: NMR solution structure of tamapin, mutant E25K/K27E 手法: SOLUTION NMR PDB-6d8u: NMR solution structure of tamapin, mutant K20E 手法: SOLUTION NMR PDB-6d8y: NMR solution structure of tamapin, mutant Y31H 手法: SOLUTION NMR PDB-6d93: NMR solution structure of tamapin, mutant Y31A 手法: SOLUTION NMR PDB-6d9o: NMR solution structure of tamapin, mutant E25A 手法: SOLUTION NMR PDB-6d9p: NMR solution structure of tamapin, mutant K27A 手法: SOLUTION NMR |
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由来 | mesobuthus tamulus (サソリ)
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キーワード | TOXIN / Tamapin mutant / DP30 / CS-alpha/beta / SK channels / Y31+N / CSalpha/beta / DP30/Y31+N / E25K / K27E / E25K/K27E / K20E / Y31H / Y31A / E25A / K27A |
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