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PDB: 4 results

7U36
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BU of 7u36 by Molmil
Crystal structure of human GSK3B in complex with ARN1484
Descriptor: (3S)-1-[(2-fluorophenoxy)acetyl]-N-(pyridin-2-yl)pyrrolidine-3-carboxamide, CHLORIDE ION, Glycogen synthase kinase-3 beta
Authors:Tripathi, S.K, Balboni, B, Giabbai, B, Storici, P, Girotto, S, Cavalli, A.
Deposit date:2022-02-25
Release date:2022-04-27
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.75 Å)
Cite:Identification of Novel GSK-3 beta Hits Using Competitive Biophysical Assays.
Int J Mol Sci, 23, 2022
7U31
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BU of 7u31 by Molmil
Crystal structure of human GSK3B in complex with G5
Descriptor: 5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amine, CHLORIDE ION, Glycogen synthase kinase-3 beta
Authors:Tripathi, S.K, Balboni, B, Giabbai, B, Storici, P, Girotto, S, Cavalli, A.
Deposit date:2022-02-25
Release date:2022-04-27
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.38 Å)
Cite:Identification of Novel GSK-3 beta Hits Using Competitive Biophysical Assays.
Int J Mol Sci, 23, 2022
7U33
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BU of 7u33 by Molmil
Crystal structure of human GSK3B in complex with ARN9133
Descriptor: 3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylazetidine-1-sulfonamide, CHLORIDE ION, Glycogen synthase kinase-3 beta
Authors:Tripathi, S.K, Balboni, B, Giabbai, B, Storici, P, Girotto, S, Cavalli, A.
Deposit date:2022-02-25
Release date:2022-04-27
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Identification of Novel GSK-3 beta Hits Using Competitive Biophysical Assays.
Int J Mol Sci, 23, 2022
7U2Z
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BU of 7u2z by Molmil
Crystal structure of human GSK3B in complex with G12
Descriptor: (3R)-1-[3-(2-fluorophenyl)propanoyl]-N-(pyridin-2-yl)pyrrolidine-3-carboxamide, CHLORIDE ION, Glycogen synthase kinase-3 beta
Authors:Tripathi, S.K, Balboni, B, Giabbai, B, Storici, P, Girotto, S, Cavalli, A.
Deposit date:2022-02-25
Release date:2022-04-27
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.21 Å)
Cite:Identification of Novel GSK-3 beta Hits Using Competitive Biophysical Assays.
Int J Mol Sci, 23, 2022

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PDB entries from 2024-05-15

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