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PDB: 4 results

7A1Y
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BU of 7a1y by Molmil
KRASG12C GDP form in complex with Cpd2
Descriptor: GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
Authors:Mathieu, M, Steier, V.
Deposit date:2020-08-14
Release date:2021-10-13
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.004 Å)
Cite:KRAS G12C fragment screening renders new binding pockets.
Small Gtpases, 13, 2022
7A1X
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BU of 7a1x by Molmil
KRASG12C GDP form in complex with Cpd1
Descriptor: 3-(imidazol-1-ylmethyl)-1~{H}-indole, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Mathieu, M, Steier, V.
Deposit date:2020-08-14
Release date:2021-10-13
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (1.32 Å)
Cite:KRAS G12C fragment screening renders new binding pockets.
Small Gtpases, 13, 2022
7A1W
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BU of 7a1w by Molmil
KRASG12C GDP form in complex with Cpd3
Descriptor: GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, MAGNESIUM ION, ...
Authors:Mathieu, M, Steier, V.
Deposit date:2020-08-14
Release date:2021-10-13
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (1.76 Å)
Cite:KRAS G12C fragment screening renders new binding pockets.
Small Gtpases, 13, 2022
7A47
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BU of 7a47 by Molmil
KRASG12C GDP form in complex with Cpd4
Descriptor: GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, ~{N}-[3-bromanyl-2-(2-methylimidazol-1-yl)pyridin-4-yl]-3-[[3-bromanyl-2-(2-methylimidazol-1-yl)pyridin-4-yl]-propanoyl-amino]propanamide
Authors:Bertrand, T, Steier, V.
Deposit date:2020-08-19
Release date:2021-10-13
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.16 Å)
Cite:KRAS G12C fragment screening renders new binding pockets.
Small Gtpases, 13, 2022

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PDB entries from 2024-05-15

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