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PDB: 4 results

6PMA
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BU of 6pma by Molmil
TRK-A IN COMPLEX WITH LIGAND
Descriptor: High affinity nerve growth factor receptor, N-[2-chloro-5-(trifluoromethyl)phenyl]-2-[1-(4-methoxyphenyl)-4-oxo-1,4-dihydro-5H-pyrazolo[3,4-d]pyrimidin-5-yl]acetamide
Authors:Subramanian, G, Brown, D.G.
Deposit date:2019-07-01
Release date:2020-02-26
Last modified:2021-02-03
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Synthetic inhibitor leads of human tropomyosin receptor kinase A ( h TrkA).
Rsc Med Chem, 11, 2020
6PMB
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BU of 6pmb by Molmil
TRK-A IN COMPLEX WITH LIGAND 1a
Descriptor: 2-[5,7-dimethyl-2-(pyridin-3-yl)[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-N-[3-(trifluoromethyl)phenyl]acetamide, High affinity nerve growth factor receptor
Authors:Subramanian, G, Brown, D.G.
Deposit date:2019-07-01
Release date:2020-02-26
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.81 Å)
Cite:Synthetic inhibitor leads of human tropomyosin receptor kinase A ( h TrkA).
Rsc Med Chem, 11, 2020
6PME
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BU of 6pme by Molmil
TRK-A IN COMPLEX WITH LIGAND
Descriptor: High affinity nerve growth factor receptor, N-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide, S,R MESO-TARTARIC ACID, ...
Authors:Subramanian, G, Brown, D.G.
Deposit date:2019-07-01
Release date:2020-02-26
Last modified:2021-02-03
Method:X-RAY DIFFRACTION (3 Å)
Cite:Synthetic inhibitor leads of human tropomyosin receptor kinase A ( h TrkA).
Rsc Med Chem, 11, 2020
6PMC
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BU of 6pmc by Molmil
TRK-A IN COMPLEX WITH LIGAND 1a
Descriptor: High affinity nerve growth factor receptor, N-(6-{[(5-chloro-2-methoxyphenyl)carbamoyl]amino}-1,3-benzothiazol-2-yl)benzamide
Authors:Subramanian, G, Brown, D.G.
Deposit date:2019-07-01
Release date:2020-02-26
Last modified:2021-02-03
Method:X-RAY DIFFRACTION (2.19 Å)
Cite:Synthetic inhibitor leads of human tropomyosin receptor kinase A ( h TrkA).
Rsc Med Chem, 11, 2020

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