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PDB: 1 results

5LHB
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POLYADPRIBOSYL GLYCOSIDASE IN COMPLEX WITH PDD00017262
Descriptor: 1-(cyclopropylmethyl)-6-[[(1-methylcyclopropyl)amino]-bis(oxidanyl)-$l^{4}-sulfanyl]-3-[(2-methyl-1,3-thiazol-5-yl)methyl]quinazoline-2,4-dione, DIMETHYL SULFOXIDE, Poly(ADP-ribose) glycohydrolase, ...
Authors:Tucker, J, Barkauskaite, E.
Deposit date:2016-07-10
Release date:2016-10-12
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.23 Å)
Cite:First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib.
ACS Chem. Biol., 11, 2016

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