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Complex structure of the first bromodomain of BRD4 with an inhibitor that containing a 2H-chromen-2-one ring
Descriptor:	Bromodomain-containing protein 4, ~{N}-methyl-~{N}-[3-[(2-oxidanylidenechromen-4-yl)amino]propyl]thiophene-2-carboxamide
Authors:	Zhang, H, Sun, Z.Y.
Deposit date:	2016-12-21
Release date:	2017-04-12
Last modified:	2023-11-22
Method:	X-RAY DIFFRACTION (1.724 Å)
Cite:	Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays. Bioorg. Med. Chem. Lett., 27, 2017