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PDB: 1 results

8FE9
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BU of 8fe9 by Molmil
Crystal structure of Ack1 kinase K161Q mutant in complex with the selective inhibitor (R)-9b
Descriptor: Activated CDC42 kinase 1, N-[(1S)-1-benzyl-2-[(6-chloro-2-oxo-1H-quinolin-4-yl)methylamino]-2-oxo-ethyl]-4-hydroxy-2-oxo-1H-quinoline-6-carbo
Authors:Paung, Y, Kan, Y, Seeliger, M.S, Miller, W.T.
Deposit date:2022-12-06
Release date:2023-03-29
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:Biochemical Studies of Systemic Lupus Erythematosus-Associated Mutations in Nonreceptor Tyrosine Kinases Ack1 and Brk.
Biochemistry, 62, 2023

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