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5ENO
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BU of 5eno by Molmil
MBX2319 bound structure of bacterial efflux pump.
Descriptor: 3,3-dimethyl-8-morpholin-4-yl-6-(2-phenylethylsulfanyl)-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrile, DARPin, Multidrug efflux pump subunit AcrB,Multidrug efflux pump subunit AcrB
Authors:Sjuts, H, Ornik, A.R, Pos, K.M.
Deposit date:2015-11-09
Release date:2016-04-06
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Molecular basis for inhibition of AcrB multidrug efflux pump by novel and powerful pyranopyridine derivatives.
Proc.Natl.Acad.Sci.USA, 113, 2016
5EN5
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BU of 5en5 by Molmil
Apo structure of bacterial efflux pump.
Descriptor: DARPin, Multidrug efflux pump subunit AcrB,Multidrug efflux pump subunit AcrB
Authors:Sjuts, H, Ornik, A.R, Pos, K.M.
Deposit date:2015-11-09
Release date:2016-04-06
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Molecular basis for inhibition of AcrB multidrug efflux pump by novel and powerful pyranopyridine derivatives.
Proc.Natl.Acad.Sci.USA, 113, 2016
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