7GTS
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![BU of 7gts by Molmil](/molmil-images/mine/7gts) | |
7GSM
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![BU of 7gsm by Molmil](/molmil-images/mine/7gsm) | |
7GTB
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![BU of 7gtb by Molmil](/molmil-images/mine/7gtb) | |
7GSO
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![BU of 7gso by Molmil](/molmil-images/mine/7gso) | |
7GTQ
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![BU of 7gtq by Molmil](/molmil-images/mine/7gtq) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOPL000311a | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1, ~{N}-(2-ethyl-1,2,3,4-tetrazol-5-yl)butanamide | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (2.09 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSX
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![BU of 7gsx by Molmil](/molmil-images/mine/7gsx) | |
7GTG
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![BU of 7gtg by Molmil](/molmil-images/mine/7gtg) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000684a | Descriptor: | (5R,7S,8R,8aS)-2-(cyclopropylmethyl)-8-phenyloctahydropyrrolo[1,2-a]pyrazine-7-carboxamide, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.69 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSU
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![BU of 7gsu by Molmil](/molmil-images/mine/7gsu) | |
7GTP
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![BU of 7gtp by Molmil](/molmil-images/mine/7gtp) | |
7GSZ
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![BU of 7gsz by Molmil](/molmil-images/mine/7gsz) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMSOA000686b | Descriptor: | 1-[4-methyl-2-(pyridin-4-yl)-1,3-thiazol-5-yl]methanamine, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.91 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GT7
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![BU of 7gt7 by Molmil](/molmil-images/mine/7gt7) | |
7GSR
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![BU of 7gsr by Molmil](/molmil-images/mine/7gsr) | |
7GTT
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![BU of 7gtt by Molmil](/molmil-images/mine/7gtt) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOPL000148a | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, N-(3,4-dihydroquinoline-1(2H)-carbothioyl)propanamide, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.93 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSV
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![BU of 7gsv by Molmil](/molmil-images/mine/7gsv) | |
7GTD
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![BU of 7gtd by Molmil](/molmil-images/mine/7gtd) | |
7GSW
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![BU of 7gsw by Molmil](/molmil-images/mine/7gsw) | |
7GTR
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![BU of 7gtr by Molmil](/molmil-images/mine/7gtr) | |
7GSQ
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![BU of 7gsq by Molmil](/molmil-images/mine/7gsq) | |
7GTE
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![BU of 7gte by Molmil](/molmil-images/mine/7gte) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with XST00000646b | Descriptor: | (5S)-5-(trifluoromethyl)-1,4-diazepane, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GTU
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![BU of 7gtu by Molmil](/molmil-images/mine/7gtu) | |
7GST
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![BU of 7gst by Molmil](/molmil-images/mine/7gst) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOMB000056a | Descriptor: | 1-(methanesulfonyl)-1,2,3,4-tetrahydroquinoline, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.64 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GT6
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![BU of 7gt6 by Molmil](/molmil-images/mine/7gt6) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000530a | Descriptor: | (3aS,8aS)-6-benzoyloctahydropyrrolo[3,4-d]azepin-1(2H)-one, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.66 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSY
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![BU of 7gsy by Molmil](/molmil-images/mine/7gsy) | |
7GTH
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![BU of 7gth by Molmil](/molmil-images/mine/7gth) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000637a | Descriptor: | (6aR,8R,12R,12aS)-2-methyl-6a,10,11,12a-tetrahydro-6H,7H,9H-[1]benzopyrano[4,3-c]pyrazolo[1,2-a]pyrazol-9-one, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.66 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSN
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![BU of 7gsn by Molmil](/molmil-images/mine/7gsn) | |