5JN2
Crystal structure of TgCDPK1 bound to NVPACU106
Summary for 5JN2
Entry DOI | 10.2210/pdb5jn2/pdb |
Related | 5JMS |
Descriptor | Calmodulin-domain protein kinase 1, N-[(3-{4-amino-5-[3-(benzyloxy)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-7-yl}cyclobutyl)methyl]acetamide, CALCIUM ION, ... (5 entities in total) |
Functional Keywords | kinase, structural genomics consortium, sgc, hydrolase |
Biological source | Toxoplasma gondii |
Total number of polymer chains | 1 |
Total formula weight | 60077.08 |
Authors | El Bakkouri, M.,Walker, J.R.,Loppnau, P.,Graslund, S.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.M.,Hui, R.,Lovato, D.V.,Structural Genomics Consortium (SGC) (deposition date: 2016-04-29, release date: 2016-05-25, Last modification date: 2023-09-27) |
Primary citation | El Bakkouri, M.,Walker, J.R.,Loppnau, P.,Graslund, S.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.M.,Hui, R.,Lovato, D.V.,Structural Genomics Consortium (SGC) Crystal structure of TgCDPK1 bound to NVPACU106 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
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