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4ZQL

Crystal structure of TRIM24 with 3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide inhibitor

Summary for 4ZQL
Entry DOI10.2210/pdb4zql/pdb
DescriptorTranscription intermediary factor 1-alpha, ZINC ION, SULFATE ION, ... (7 entities in total)
Functional Keywordstranscriptional coactivator, histone h3 modifications, e3 protein-ubiquitin ligase activity, structural genomics, structural genomics consortium, sgc, ligase
Biological sourceHomo sapiens (Human)
Cellular locationNucleus : O15164
Total number of polymer chains2
Total formula weight44076.80
Authors
Primary citationClark, P.G.,Vieira, L.C.,Tallant, C.,Fedorov, O.,Singleton, D.C.,Rogers, C.M.,Monteiro, O.P.,Bennett, J.M.,Baronio, R.,Muller, S.,Daniels, D.L.,Mendez, J.,Knapp, S.,Brennan, P.E.,Dixon, D.J.
Crystal structure of TRIM24 with 3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.79 Å)
Structure validation

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PDB entries from 2024-03-27

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