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3VJS

Vitamin D receptor complex with a carborane compound

Summary for 3VJS
Entry DOI10.2210/pdb3vjs/pdb
Related3VJT
DescriptorVitamin D3 receptor, peptide from Mediator of RNA polymerase II transcription subunit 1, 1-(2-[(S)-2,4-Dihydroxybutoxy]ethyl)-12-(5-ethyl-5-hydroxyheptyl)-1,12-dicarba-closo-dodecaborane, ... (4 entities in total)
Functional Keywordsnuclear receptor, synthetic agonist, carborane, transcription
Biological sourceRattus norvegicus (Rat)
More
Cellular locationNucleus: P13053 Q15648
Total number of polymer chains2
Total formula weight32584.56
Authors
Fujii, S.,Masuno, M.,Kagechika, H.,Nakabayashi, M.,Ito, N. (deposition date: 2011-10-31, release date: 2012-02-08, Last modification date: 2023-11-08)
Primary citationFujii, S.,Masuno, H.,Taoda, Y.,Kano, A.,Wongmayura, A.,Nakabayashi, M.,Ito, N.,Shimizu, M.,Kawachi, E.,Hirano, T.,Endo, Y.,Tanatani, A.,Kagechika, H.
Boron Cluster-based Development of Potent Nonsecosteroidal Vitamin D Receptor Ligands: Direct Observation of Hydrophobic Interaction between Protein Surface and Carborane
J.Am.Chem.Soc., 133:20933-20941, 2011
Cited by
PubMed: 22066785
DOI: 10.1021/ja208797n
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.93 Å)
Structure validation

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