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7F59
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BU of 7f59 by Molmil
DNQX-bound GluK2-1xNeto2 complex
Descriptor: (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (4.2 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F56
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BU of 7f56 by Molmil
DNQX-bound GluK2-1xNeto2 complex, with asymmetric LBD
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (4.1 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F5B
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BU of 7f5b by Molmil
LBD-TMD focused reconstruction of DNQX-bound GluK2-1xNeto2 complex
Descriptor: (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (3.9 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F57
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BU of 7f57 by Molmil
Kainate-bound GluK2-1xNeto2 complex, at the desensitized state
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (3.8 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F5A
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BU of 7f5a by Molmil
DNQX-bound GluK2-2xNeto2 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (6.4 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
8R36
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BU of 8r36 by Molmil
Crystal structure of the Gluk1 ligand-binding domain in complex with kainate and BPAM538 at 1.90 A resolution
Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, 4-cyclopropyl-7-(3-methoxyphenoxy)-2,3-dihydro-1$l^{6},2,4-benzothiadiazine 1,1-dioxide, CHLORIDE ION, ...
Authors:Bay, Y, Frantsen, S.M, Frydenvang, K, Kastrup, J.S.
Deposit date:2023-11-08
Release date:2024-08-14
Last modified:2024-09-04
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystal structure of the GluK1 ligand-binding domain with kainate and the full-spanning positive allosteric modulator BPAM538.
J.Struct.Biol., 216, 2024

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PDB entries from 2024-09-18

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