登録情報 データベース : PDB / ID : 8qzd 構造の表示 ダウンロードとリンクタイトル Soluble epoxide hydrolase in complex with Epoxykinin 要素Bifunctional epoxide hydrolase 2 詳細 キーワード HYDROLASE / COMPLEX / STRUCTURAL GENOMICS / STRUCTURAL GENOMICS CONSORTIUM / SGC機能・相同性 機能・相同性情報分子機能 ドメイン・相同性 構成要素
lipid-phosphate phosphatase / 10-hydroxy-9-(phosphonooxy)octadecanoate phosphatase activity / stilbene catabolic process / Biosynthesis of maresins / phospholipid dephosphorylation / soluble epoxide hydrolase / epoxide metabolic process / lipid phosphatase activity / lysophosphatidic acid phosphatase activity / Synthesis of epoxy (EET) and dihydroxyeicosatrienoic acids (DHET) ... lipid-phosphate phosphatase / 10-hydroxy-9-(phosphonooxy)octadecanoate phosphatase activity / stilbene catabolic process / Biosynthesis of maresins / phospholipid dephosphorylation / soluble epoxide hydrolase / epoxide metabolic process / lipid phosphatase activity / lysophosphatidic acid phosphatase activity / Synthesis of epoxy (EET) and dihydroxyeicosatrienoic acids (DHET) / epoxide hydrolase activity / regulation of cholesterol metabolic process / phosphatase activity / peroxisomal matrix / toxic substance binding / dephosphorylation / cholesterol homeostasis / Peroxisomal protein import / response to toxic substance / peroxisome / positive regulation of gene expression / magnesium ion binding / protein homodimerization activity / extracellular exosome / cytosol 類似検索 - 分子機能 Predicted HAD-superfamily phosphatase, subfamily IA/Epoxide hydrolase, N-terminal / Phosphoglycolate phosphatase-like, domain 2 / HAD hydrolase, subfamily IA / Epoxide hydrolase-like / alpha/beta hydrolase fold / haloacid dehalogenase-like hydrolase / Alpha/beta hydrolase fold-1 / HAD superfamily / HAD-like superfamily / Alpha/Beta hydrolase fold 類似検索 - ドメイン・相同性 BROMIDE ION / : / Bifunctional epoxide hydrolase 2 類似検索 - 構成要素生物種 Homo sapiens (ヒト)手法 X線回折 / シンクロトロン / 分子置換 / 解像度 : 1.3 Å 詳細データ登録者 Kumar, A. / Ehrler, J.M.H. / Ziegler, S. / Doetsch, L. / Proschak, E. / Knapp, S. / Structural Genomics Consortium (SGC) 資金援助 European Union, スイス, 3件 詳細 詳細を隠す組織 認可番号 国 European Union (EU) EFRE-0200481 European Union Innovative Medicines Initiative 115489 スイス European Communitys Seventh Framework Programme FP7/2007-2013 European Union
引用ジャーナル : J.Med.Chem. / 年 : 2024タイトル : Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator.著者 : Dotsch, L. / Davies, C. / Hennes, E. / Schonfeld, J. / Kumar, A. / Guita, C.D.C.L. / Ehrler, J.H.M. / Hiesinger, K. / Thavam, S. / Janning, P. / Sievers, S. / Knapp, S. / Proschak, E. / Ziegler, S. / Waldmann, H. 履歴 登録 2023年10月27日 登録サイト : PDBE / 処理サイト : PDBE改定 1.0 2024年2月28日 Provider : repository / タイプ : Initial release改定 1.1 2024年4月3日 Group : Database references / カテゴリ : citation / citation_authorItem : _citation.country / _citation.journal_abbrev ... _citation.country / _citation.journal_abbrev / _citation.journal_id_ASTM / _citation.journal_id_CSD / _citation.journal_id_ISSN / _citation.journal_volume / _citation.page_first / _citation.page_last / _citation.pdbx_database_id_DOI / _citation.pdbx_database_id_PubMed / _citation.title / _citation.year
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