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-Structure paper
Title | Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator. |
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Journal, issue, pages | J. Med. Chem., Vol. 67, Page 4691-4706, Year 2024 |
Publish date | Oct 27, 2023 (structure data deposition date) |
Authors | Dotsch, L. / Davies, C. / Hennes, E. / Schonfeld, J. / Kumar, A. / Guita, C.D.C.L. / Ehrler, J.H.M. / Hiesinger, K. / Thavam, S. / Janning, P. ...Dotsch, L. / Davies, C. / Hennes, E. / Schonfeld, J. / Kumar, A. / Guita, C.D.C.L. / Ehrler, J.H.M. / Hiesinger, K. / Thavam, S. / Janning, P. / Sievers, S. / Knapp, S. / Proschak, E. / Ziegler, S. / Waldmann, H. |
External links | J. Med. Chem. / PubMed:38470246 |
Methods | X-ray diffraction |
Resolution | 1.3 Å |
Structure data | PDB-8qzd: |
Chemicals | ChemComp-EDO:
ChemComp-XDZ: ChemComp-BR: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / COMPLEX / STRUCTURAL GENOMICS / STRUCTURAL GENOMICS CONSORTIUM / SGC |