登録情報 | データベース: PDB / ID: 8cgz |
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タイトル | tubulin-AB8939 complex |
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要素 | - Stathmin-4
- Tubulin alpha chain
- Tubulin beta chain
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キーワード | CELL CYCLE / MICROTUBULE DYNAMICS / INHIBITOR / CYTOSKELETON / CELL DIVISION |
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機能・相同性 | 機能・相同性情報
axonemal microtubule / organelle transport along microtubule / glial cell differentiation / forebrain morphogenesis / neuron projection arborization / cerebellar cortex morphogenesis / dentate gyrus development / pyramidal neuron differentiation / centrosome cycle / motor behavior ...axonemal microtubule / organelle transport along microtubule / glial cell differentiation / forebrain morphogenesis / neuron projection arborization / cerebellar cortex morphogenesis / dentate gyrus development / pyramidal neuron differentiation / centrosome cycle / motor behavior / microtubule depolymerization / response to L-glutamate / smoothened signaling pathway / regulation of synapse organization / startle response / locomotory exploration behavior / microtubule polymerization / regulation of microtubule polymerization or depolymerization / response to tumor necrosis factor / response to mechanical stimulus / condensed chromosome / homeostasis of number of cells within a tissue / cellular response to calcium ion / tubulin binding / adult locomotory behavior / intracellular protein transport / neuron migration / synapse organization / visual learning / neuromuscular junction / recycling endosome / cerebral cortex development / structural constituent of cytoskeleton / memory / microtubule cytoskeleton organization / cytoplasmic ribonucleoprotein granule / neuron projection development / mitotic cell cycle / gene expression / growth cone / neuron apoptotic process / microtubule / hydrolase activity / neuron projection / protein heterodimerization activity / GTPase activity / GTP binding / protein-containing complex binding / Golgi apparatus / identical protein binding / metal ion binding / plasma membrane / cytosol / cytoplasm類似検索 - 分子機能 Stathmin family / Stathmin, conserved site / Stathmin superfamily / Stathmin family / Stathmin family signature 1. / Stathmin family signature 2. / Stathmin-like (SLD) domain profile. / Alpha tubulin / Tubulin-beta mRNA autoregulation signal. / Beta tubulin, autoregulation binding site ...Stathmin family / Stathmin, conserved site / Stathmin superfamily / Stathmin family / Stathmin family signature 1. / Stathmin family signature 2. / Stathmin-like (SLD) domain profile. / Alpha tubulin / Tubulin-beta mRNA autoregulation signal. / Beta tubulin, autoregulation binding site / Beta tubulin / Tubulin / Tubulin, C-terminal / Tubulin C-terminal domain / Tubulin, conserved site / Tubulin subunits alpha, beta, and gamma signature. / Tubulin/FtsZ family, C-terminal domain / Tubulin/FtsZ-like, C-terminal domain / Tubulin/FtsZ, C-terminal / Tubulin/FtsZ, 2-layer sandwich domain / Tubulin/FtsZ family, GTPase domain / Tubulin/FtsZ family, GTPase domain / Tubulin/FtsZ, GTPase domain / Tubulin/FtsZ, GTPase domain superfamily類似検索 - ドメイン・相同性 GUANOSINE-5'-DIPHOSPHATE / GUANOSINE-5'-TRIPHOSPHATE / : / Tubulin beta chain / Tubulin alpha chain / Stathmin-4類似検索 - 構成要素 |
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生物種 | Rattus norvegicus (ドブネズミ) Ovis aries (ヒツジ) |
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手法 | X線回折 / シンクロトロン / フーリエ合成 / 解像度: 2.527 Å |
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データ登録者 | Varela, P.F. / Gigant, B. |
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資金援助 | フランス, 1件 組織 | 認可番号 | 国 |
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Fondation ARC | ARCPJA2021050003651 | フランス |
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引用 | ジャーナル: TO BE PUBLISHED タイトル: Development of AB8939, a Novel Colchicine-like Microtubule Synthetic Destabilizer with the Ability to Overcome Multidrug Resistance 著者: Humbert, M. / Letard, S. / Neves, M. / Siavoshian Jeay, S. / Goubard, A. / Casteran, N. / Rebuffet, E. / Hajem, B. / Gros, L. / Varela, P.F. / Gigant, B. / Verdier, P. / Castellano, R. / ...著者: Humbert, M. / Letard, S. / Neves, M. / Siavoshian Jeay, S. / Goubard, A. / Casteran, N. / Rebuffet, E. / Hajem, B. / Gros, L. / Varela, P.F. / Gigant, B. / Verdier, P. / Castellano, R. / Colette, Y. / Vey, N. / Pez, D. / Benjahad, A. / Moussy, A. / Mansfield, C. / Dubreuil, P. |
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履歴 | 登録 | 2023年2月6日 | 登録サイト: PDBE / 処理サイト: PDBE |
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改定 1.0 | 2024年8月14日 | Provider: repository / タイプ: Initial release |
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