登録情報 データベース : PDB / ID : 2yjd 構造の表示 ダウンロードとリンクタイトル Stapled peptide bound to Estrogen Receptor Beta 要素ESTROGEN RECEPTOR BETA STAPLED PEPTIDE 詳細キーワード HORMONE RECEPTOR/PEPTIDE / HORMONE RECEPTOR-PEPTIDE COMPLEX機能・相同性 機能・相同性情報分子機能 ドメイン・相同性 構成要素
receptor antagonist activity / nuclear steroid receptor activity / RNA polymerase II intronic transcription regulatory region sequence-specific DNA binding / nuclear estrogen receptor activity / locomotor rhythm / aryl hydrocarbon receptor binding / regulation of lipid metabolic process / cellular response to Thyroglobulin triiodothyronine / regulation of glucose metabolic process / Synthesis of bile acids and bile salts ... receptor antagonist activity / nuclear steroid receptor activity / RNA polymerase II intronic transcription regulatory region sequence-specific DNA binding / nuclear estrogen receptor activity / locomotor rhythm / aryl hydrocarbon receptor binding / regulation of lipid metabolic process / cellular response to Thyroglobulin triiodothyronine / regulation of glucose metabolic process / Synthesis of bile acids and bile salts / estrogen receptor signaling pathway / cellular response to estrogen stimulus / positive regulation of adipose tissue development / peroxisome proliferator activated receptor signaling pathway / Endogenous sterols / Synthesis of bile acids and bile salts via 27-hydroxycholesterol / estrogen response element binding / Synthesis of bile acids and bile salts via 7alpha-hydroxycholesterol / regulation of cellular response to insulin stimulus / Recycling of bile acids and salts / cellular response to hormone stimulus / cellular response to estradiol stimulus / RORA activates gene expression / steroid binding / Regulation of lipid metabolism by PPARalpha / ESR-mediated signaling / BMAL1:CLOCK,NPAS2 activates circadian gene expression / SUMOylation of transcription cofactors / Activation of gene expression by SREBF (SREBP) / nuclear receptor coactivator activity / mRNA transcription by RNA polymerase II / response to progesterone / nuclear receptor binding / PPARA activates gene expression / positive regulation of DNA-binding transcription factor activity / circadian regulation of gene expression / Heme signaling / Activated PKN1 stimulates transcription of AR (androgen receptor) regulated genes KLK2 and KLK3 / Nuclear Receptor transcription pathway / Transcriptional activation of mitochondrial biogenesis / Transcriptional regulation of white adipocyte differentiation / Cytoprotection by HMOX1 / negative regulation of cell growth / RNA polymerase II transcription regulator complex / Constitutive Signaling by Aberrant PI3K in Cancer / nuclear receptor activity / PIP3 activates AKT signaling / Circadian Clock / cell-cell signaling / PI5P, PP2A and IER3 Regulate PI3K/AKT Signaling / HATs acetylate histones / transcription regulator complex / Estrogen-dependent gene expression / transcription coactivator activity / Extra-nuclear estrogen signaling / DNA-binding transcription factor activity, RNA polymerase II-specific / protein dimerization activity / nuclear body / RNA polymerase II cis-regulatory region sequence-specific DNA binding / protein domain specific binding / intracellular membrane-bounded organelle / chromatin binding / regulation of transcription by RNA polymerase II / positive regulation of DNA-templated transcription / chromatin / regulation of DNA-templated transcription / enzyme binding / negative regulation of transcription by RNA polymerase II / signal transduction / positive regulation of transcription by RNA polymerase II / protein-containing complex / mitochondrion / DNA binding / zinc ion binding / nucleoplasm / nucleus / cytoplasm 類似検索 - 分子機能 Estrogen receptor beta-like, N-terminal / Estrogen receptor beta/gamma / Estrogen receptor beta / Nuclear receptor coactivator 2 / Nuclear receptor coactivator 2/3, DUF4927 / Domain of unknown function (DUF4927) / Estrogen receptor/oestrogen-related receptor / Nuclear receptor coactivator, DUF1518 / Nuclear receptor coactivator, Ncoa-type, interlocking / Nuclear receptor coactivator, Ncoa-type, interlocking domain superfamily ... Estrogen receptor beta-like, N-terminal / Estrogen receptor beta/gamma / Estrogen receptor beta / Nuclear receptor coactivator 2 / Nuclear receptor coactivator 2/3, DUF4927 / Domain of unknown function (DUF4927) / Estrogen receptor/oestrogen-related receptor / Nuclear receptor coactivator, DUF1518 / Nuclear receptor coactivator, Ncoa-type, interlocking / Nuclear receptor coactivator, Ncoa-type, interlocking domain superfamily / Nuclear receptor coactivator, DUF1518 / Nuclear receptor coactivator / DUF1518 / Nuclear receptor coactivator, receptor-binding domain / Nuclear receptor coactivator / Steroid receptor coactivator / Unstructured region on nuclear receptor coactivator protein / PAS domain / : / Nuclear receptor coactivator, interlocking / Helix-loop-helix DNA-binding domain superfamily / helix loop helix domain / Myc-type, basic helix-loop-helix (bHLH) domain / Myc-type, basic helix-loop-helix (bHLH) domain profile. / PAS fold / PAS fold / PAS domain / PAS repeat profile. / PAS domain / Retinoid X Receptor / Retinoid X Receptor / PAS domain superfamily / Nuclear hormone receptor / Nuclear hormones receptors DNA-binding region signature. / Zinc finger, nuclear hormone receptor-type / Zinc finger, C4 type (two domains) / Nuclear hormone receptors DNA-binding domain profile. / c4 zinc finger in nuclear hormone receptors / Nuclear hormone receptor, ligand-binding domain / Nuclear hormone receptor-like domain superfamily / Nuclear receptor (NR) ligand-binding (LBD) domain profile. / Ligand binding domain of hormone receptors / Zinc finger, NHR/GATA-type / Ligand-binding domain of nuclear hormone receptor / Orthogonal Bundle / Mainly Alpha 類似検索 - ドメイン・相同性 4-(2-PROPAN-2-YLOXYBENZIMIDAZOL-1-YL)PHENOL / Nuclear receptor coactivator 2 / Estrogen receptor beta 類似検索 - 構成要素生物種 HOMO SAPIENS (ヒト)手法 X線回折 / OTHER / 解像度 : 1.93 Å 詳細データ登録者 Phillips, C. / Roberts, L.R. / Schade, M. / Bent, A. / Davies, N.L. / Moore, R. / Pannifer, A.D. / Brown, D.G. / Pickford, A.R. / Irving, S.L. 引用ジャーナル : J.Am.Chem.Soc. / 年 : 2011タイトル : Design and Structure of Stapled Peptides Binding to Estrogen Receptors.著者 : Phillips, C. / Roberts, L.R. / Schade, M. / Bazin, R. / Bent, A. / Davies, N.L. / Moore, R. / Pannifer, A.D. / Pickford, A.R. / Prior, S.H. / Read, C.M. / Scott, A. / Brown, D.G. / Xu, B. / Irving, S.L. 履歴 登録 2011年5月19日 登録サイト : PDBE / 処理サイト : PDBE改定 1.0 2011年8月3日 Provider : repository / タイプ : Initial release改定 1.1 2017年1月25日 Group : Atomic model / Other
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