Mass: 18.015 Da / Num. of mol.: 293 / Source method: isolated from a natural source / Formula: H2O
Compound details
CASEIN KINASES ARE OPERATIONALLY DEFINED BY THEIR PREFERENTIAL UTILIZATION OF ACIDIC PROTEINS SUCH ...CASEIN KINASES ARE OPERATIONALLY DEFINED BY THEIR PREFERENTIAL UTILIZATION OF ACIDIC PROTEINS SUCH AS CASEINS AS SUBSTRATES. IT CAN PHOSPHORYLATE A LARGE NUMBER OF PROTEINS.
Sequence details
NTERMINAL SER-MET ARE DERIVED FROM CLONING
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Experimental details
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Experiment
Experiment
Method: X-RAY DIFFRACTION / Number of used crystals: 1
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Sample preparation
Crystal
Density Matthews: 2.57 Å3/Da / Density % sol: 52 %
Resolution: 1.75→50 Å / Cor.coef. Fo:Fc: 0.968 / Cor.coef. Fo:Fc free: 0.947 / SU B: 4.147 / SU ML: 0.075 / TLS residual ADP flag: LIKELY RESIDUAL / Cross valid method: THROUGHOUT / ESU R: 0.098 / ESU R Free: 0.101 / Stereochemistry target values: MAXIMUM LIKELIHOOD Details: HYDROGENS HAVE BEEN ADDED IN THE RIDING POSITIONS. DIETHYLAMINO TAIL OF LIGAND IS DISORDERED AND HAS NOT BEEN INCLUDED IN THE FINAL MODEL
Rfactor
Num. reflection
% reflection
Selection details
Rfree
0.204
1914
5 %
RANDOM
Rwork
0.165
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obs
0.167
36288
99.8 %
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Solvent computation
Ion probe radii: 0.8 Å / Shrinkage radii: 0.8 Å / VDW probe radii: 1.2 Å / Solvent model: BABINET MODEL WITH MASK