- PDB-7oe9: C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH rac-N5-((1R,5S)-3-oxabi... -
+
データを開く
IDまたはキーワード:
読み込み中...
-
基本情報
登録情報
データベース: PDB / ID: 7oe9
タイトル
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH rac-N5-((1R,5S)-3-oxabicyclo[3.1.0]hexan-6-yl)-N7,3-dimethyl-3-phenyl-2,3-dihydrobenzofuran-5,7-dicarboxamide
要素
Bromodomain-containing protein 2
キーワード
NUCLEAR PROTEIN / Inhibitor / Bromodomain
機能・相同性
機能・相同性情報
acetylation-dependent protein binding / chromatin looping / RUNX3 regulates p14-ARF / positive regulation of T-helper 17 cell lineage commitment / protein localization to chromatin / neural tube closure / lysine-acetylated histone binding / nucleosome assembly / spermatogenesis / nuclear speck ...acetylation-dependent protein binding / chromatin looping / RUNX3 regulates p14-ARF / positive regulation of T-helper 17 cell lineage commitment / protein localization to chromatin / neural tube closure / lysine-acetylated histone binding / nucleosome assembly / spermatogenesis / nuclear speck / protein serine/threonine kinase activity / chromatin binding / chromatin / regulation of transcription by RNA polymerase II / nucleoplasm / nucleus / cytoplasm 類似検索 - 分子機能
NET domain superfamily / NET domain profile. / Brdt, bromodomain, repeat II / Brdt, bromodomain, repeat I / : / NET domain / Bromodomain extra-terminal - transcription regulation / Bromodomain, conserved site / Bromodomain signature. / Bromodomain ...NET domain superfamily / NET domain profile. / Brdt, bromodomain, repeat II / Brdt, bromodomain, repeat I / : / NET domain / Bromodomain extra-terminal - transcription regulation / Bromodomain, conserved site / Bromodomain signature. / Bromodomain / Bromodomain profile. / bromo domain / Bromodomain / Bromodomain-like superfamily 類似検索 - ドメイン・相同性
Chem-V9N / Bromodomain-containing protein 2 類似検索 - 構成要素
プロトコル: SINGLE WAVELENGTH / 単色(M)・ラウエ(L): M / 散乱光タイプ: x-ray
放射波長
波長: 1.54178 Å / 相対比: 1
反射
解像度: 1.6→52.45 Å / Num. obs: 14973 / % possible obs: 90.3 % / 冗長度: 2.8 % / CC1/2: 0.997 / Rmerge(I) obs: 0.024 / Net I/σ(I): 24.1
反射 シェル
解像度: 1.6→1.69 Å / 冗長度: 2 % / Rmerge(I) obs: 0.185 / Mean I/σ(I) obs: 4.7 / Num. unique obs: 1679 / CC1/2: 0.754 / % possible all: 71.5
-
解析
ソフトウェア
名称
バージョン
分類
BUSTER
2.11.7 (6-FEB-2020)
精密化
XDS
データ削減
Aimless
データスケーリング
精密化
構造決定の手法: フーリエ合成 開始モデル: in house 解像度: 1.602→14.12 Å / Cor.coef. Fo:Fc: 0.953 / Cor.coef. Fo:Fc free: 0.943 / SU R Cruickshank DPI: 0.095 / 交差検証法: THROUGHOUT / SU R Blow DPI: 0.105 / SU Rfree Blow DPI: 0.096 / SU Rfree Cruickshank DPI: 0.09