登録情報 | データベース: PDB / ID: 6p9e |
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タイトル | Crystal structure of IL-36gamma complexed to A-552 |
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要素 | Interleukin-36 gamma |
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キーワード | CYTOKINE / IL-36 / small molecule antagonist |
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機能・相同性 | 機能・相同性情報
Interleukin-36 pathway / interleukin-1 receptor binding / inflammatory response to antigenic stimulus / cytokine activity / cytokine-mediated signaling pathway / cell-cell signaling / cellular response to lipopolysaccharide / innate immune response / positive regulation of gene expression / extracellular space ...Interleukin-36 pathway / interleukin-1 receptor binding / inflammatory response to antigenic stimulus / cytokine activity / cytokine-mediated signaling pathway / cell-cell signaling / cellular response to lipopolysaccharide / innate immune response / positive regulation of gene expression / extracellular space / extracellular region / nucleoplasm / plasma membrane / cytosol類似検索 - 分子機能 Interleukin-1 receptor antagonist/Interleukin-36 / Interleukin-1 homologues / Interleukin-1 family / Interleukin-1 / 18 / Cytokine IL1/FGF / Trefoil (Acidic Fibroblast Growth Factor, subunit A) - #50 / Trefoil (Acidic Fibroblast Growth Factor, subunit A) / Trefoil / Mainly Beta類似検索 - ドメイン・相同性 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 2 Å |
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データ登録者 | Argiriadi, M.A. / Todorovic, T. / Su, Z. / Putman, B. / Kakavas, S.J. / Salte, K.M. / McDonald, H.A. / Wetter, J.B. / Paulsboe, S.E. / Sun, Q. ...Argiriadi, M.A. / Todorovic, T. / Su, Z. / Putman, B. / Kakavas, S.J. / Salte, K.M. / McDonald, H.A. / Wetter, J.B. / Paulsboe, S.E. / Sun, Q. / Gerstein, C.E. / Medina, L. / Sielaff, B. / Sadhukhan, R. / Stockmann, H. / Richardson, P.L. / Qiu, W. / Henry, R.F. / Herold, J.M. / Shotwell, J.B. / McGaraughty, S.P. / Honore, P. / Gopalakrishnan, S.M. / Sun, C.C. / Scott, V.E. |
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引用 | ジャーナル: Sci Rep / 年: 2019 タイトル: Small Molecule IL-36 gamma Antagonist as a Novel Therapeutic Approach for Plaque Psoriasis. 著者: Todorovic, V. / Su, Z. / Putman, C.B. / Kakavas, S.J. / Salte, K.M. / McDonald, H.A. / Wetter, J.B. / Paulsboe, S.E. / Sun, Q. / Gerstein, C.E. / Medina, L. / Sielaff, B. / Sadhukhan, R. / ...著者: Todorovic, V. / Su, Z. / Putman, C.B. / Kakavas, S.J. / Salte, K.M. / McDonald, H.A. / Wetter, J.B. / Paulsboe, S.E. / Sun, Q. / Gerstein, C.E. / Medina, L. / Sielaff, B. / Sadhukhan, R. / Stockmann, H. / Richardson, P.L. / Qiu, W. / Argiriadi, M.A. / Henry, R.F. / Herold, J.M. / Shotwell, J.B. / McGaraughty, S.P. / Honore, P. / Gopalakrishnan, S.M. / Sun, C.C. / Scott, V.E. |
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履歴 | 登録 | 2019年6月10日 | 登録サイト: RCSB / 処理サイト: RCSB |
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改定 1.0 | 2019年6月26日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2019年7月10日 | Group: Data collection / Database references / カテゴリ: citation / citation_author Item: _citation.country / _citation.journal_abbrev ..._citation.country / _citation.journal_abbrev / _citation.journal_id_CSD / _citation.journal_id_ISSN / _citation.journal_volume / _citation.page_first / _citation.page_last / _citation.pdbx_database_id_DOI / _citation.pdbx_database_id_PubMed / _citation.title / _citation.year / _citation_author.identifier_ORCID / _citation_author.name |
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改定 1.2 | 2023年10月11日 | Group: Data collection / Database references / Refinement description カテゴリ: chem_comp_atom / chem_comp_bond ...chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model / software Item: _database_2.pdbx_DOI / _database_2.pdbx_database_accession / _software.name |
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