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-Structure paper
Title | Covalent Modifier Discovery Using Hydrogen/Deuterium Exchange-Mass Spectrometry. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 4827-4839, Year 2023 |
Publish date | Nov 16, 2022 (structure data deposition date) |
Authors | Kojima, H. / Yanagi, R. / Higuchi, E. / Yoshizawa, M. / Shimodaira, T. / Kumagai, M. / Kyoya, T. / Sekine, M. / Egawa, D. / Ohashi, N. ...Kojima, H. / Yanagi, R. / Higuchi, E. / Yoshizawa, M. / Shimodaira, T. / Kumagai, M. / Kyoya, T. / Sekine, M. / Egawa, D. / Ohashi, N. / Ishida, H. / Yamamoto, K. / Itoh, T. |
External links | J. Med. Chem. / PubMed:36994595 |
Methods | X-ray diffraction |
Resolution | 2.4 - 2.45 Å |
Structure data | PDB-8hhp: PDB-8hhq: |
Chemicals | ChemComp-NZA: ChemComp-LRG: ChemComp-HOH: ChemComp-GOA: |
Source |
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Keywords | TRANSCRIPTION / PPARg-LBD / Partial agonists / nTZDpa / LT175 / Iodoacetic acid / Cysteine / Covalent modifier |