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Title | Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314. |
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Journal, issue, pages | Acs Pharmacol Transl Sci, Vol. 5, Page 20-40, Year 2022 |
Publish date | Jul 29, 2021 (structure data deposition date) |
![]() | Bresinsky, M. / Strasser, J.M. / Vallaster, B. / Liu, P. / McCue, W.M. / Fuller, J. / Hubmann, A. / Singh, G. / Nelson, K.M. / Cuellar, M.E. ...Bresinsky, M. / Strasser, J.M. / Vallaster, B. / Liu, P. / McCue, W.M. / Fuller, J. / Hubmann, A. / Singh, G. / Nelson, K.M. / Cuellar, M.E. / Wilmot, C.M. / Finzel, B.C. / Ashe, K.H. / Walters, M.A. / Pockes, S. |
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Methods | X-ray diffraction |
Resolution | 1.67 - 3.25 Å |
Structure data | ![]() PDB-7rn7: ![]() PDB-7rn8: ![]() PDB-7rn9: ![]() PDB-7rnb: ![]() PDB-7rnd: ![]() PDB-7rne: ![]() PDB-7rnf: ![]() PDB-7seo: |
Chemicals | ![]() ChemComp-HOH: |
Source |
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![]() | Hydrolase/Hydrolase Inhibitor / HYDROLASE / Hydrolase-Hydrolase Inhibitor complex / APOPTOSIS / protease / inhibitor / covalent |