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Title | Scaffold-Hopping Approach To Discover Potent, Selective, and Efficacious Inhibitors of NF-kappa B Inducing Kinase. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 6801-6813, Year 2018 |
Publish date | Mar 28, 2018 (structure data deposition date) |
Authors | Blaquiere, N. / Castanedo, G.M. / Burch, J.D. / Berezhkovskiy, L.M. / Brightbill, H. / Brown, S. / Chan, C. / Chiang, P.C. / Crawford, J.J. / Dong, T. ...Blaquiere, N. / Castanedo, G.M. / Burch, J.D. / Berezhkovskiy, L.M. / Brightbill, H. / Brown, S. / Chan, C. / Chiang, P.C. / Crawford, J.J. / Dong, T. / Fan, P. / Feng, J. / Ghilardi, N. / Godemann, R. / Gogol, E. / Grabbe, A. / Hole, A.J. / Hu, B. / Hymowitz, S.G. / Alaoui Ismaili, M.H. / Le, H. / Lee, P. / Lee, W. / Lin, X. / Liu, N. / McEwan, P.A. / McKenzie, B. / Silvestre, H.L. / Suto, E. / Sujatha-Bhaskar, S. / Wu, G. / Wu, L.C. / Zhang, Y. / Zhong, Z. / Staben, S.T. |
External links | J. Med. Chem. / PubMed:29940120 |
Methods | X-ray diffraction |
Resolution | 2.65 - 2.84 Å |
Structure data | PDB-6g4y: PDB-6g4z: |
Chemicals | ChemComp-SO4: ChemComp-ELZ: ChemComp-HOH: ChemComp-ELW: |
Source |
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Keywords | TRANSFERASE / PROTEIN SERINE/THREONINE KINASE / NF-KAPPAB / MAP3K14 |