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-Structure paper
Title | Conversion of Bim-BH3 from Activator to Inhibitor of Bak through Structure-Based Design. |
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Journal, issue, pages | Mol. Cell, Vol. 68, Page 659-672.e9, Year 2017 |
Publish date | May 23, 2017 (structure data deposition date) |
![]() | Brouwer, J.M. / Lan, P. / Cowan, A.D. / Bernardini, J.P. / Birkinshaw, R.W. / van Delft, M.F. / Sleebs, B.E. / Robin, A.Y. / Wardak, A. / Tan, I.K. ...Brouwer, J.M. / Lan, P. / Cowan, A.D. / Bernardini, J.P. / Birkinshaw, R.W. / van Delft, M.F. / Sleebs, B.E. / Robin, A.Y. / Wardak, A. / Tan, I.K. / Reljic, B. / Lee, E.F. / Fairlie, W.D. / Call, M.J. / Smith, B.J. / Dewson, G. / Lessene, G. / Colman, P.M. / Czabotar, P.E. |
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Methods | X-ray diffraction |
Resolution | 1.224 - 2.802 Å |
Structure data | ![]() PDB-5vwv: ![]() PDB-5vww: ![]() PDB-5vwx: ![]() PDB-5vwy: ![]() PDB-5vwz: ![]() PDB-5vx0: ![]() PDB-5vx1: ![]() PDB-5vx2: ![]() PDB-5vx3: |
Chemicals | ![]() ChemComp-TFA: ![]() ChemComp-EDO: ![]() ChemComp-CL: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-MPD: ![]() ChemComp-BR: ![]() ChemComp-IMD: ![]() ChemComp-PO4: ![]() ChemComp-1PG: ![]() ChemComp-NH4: ![]() ChemComp-MG: |
Source |
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![]() | APOPTOSIS / Bcl-2 Family / Activator / Inhibitor / Mutant / Pro-surivial / Pro-survival |