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-Structure paper
Title | Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 1876-1891, Year 2017 |
Publish date | Nov 3, 2016 (structure data deposition date) |
Authors | Xiong, Y. / Li, F. / Babault, N. / Dong, A. / Zeng, H. / Wu, H. / Chen, X. / Arrowsmith, C.H. / Brown, P.J. / Liu, J. ...Xiong, Y. / Li, F. / Babault, N. / Dong, A. / Zeng, H. / Wu, H. / Chen, X. / Arrowsmith, C.H. / Brown, P.J. / Liu, J. / Vedadi, M. / Jin, J. |
External links | J. Med. Chem. / PubMed:28135087 |
Methods | X-ray diffraction |
Resolution | 1.66 - 2.6 Å |
Structure data | PDB-5ttf: PDB-5ttg: PDB-5tuy: PDB-5tuz: |
Chemicals | ChemComp-ZN: ChemComp-SAM: ChemComp-7KZ: ChemComp-CL: ChemComp-UNX: ChemComp-HOH: ChemComp-GOL: ChemComp-DMS: ChemComp-7L6: ChemComp-EDO: |
Source |
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Keywords | TRANSFERASE / EHMT2 / G9a / BAT8 / methyltransferase / UNC3832 / Structural Genomics / Structural Genomics Consortium / SGC / EHMT1 / GLP / MS012 / TRANSFERASE/TRANSFERASE INHIBITOR / Methyl-TRANSFERASE INHIBITOR complex / TRANSFERASE-TRANSFERASE INHIBITOR complex / Methyl Transferase |