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-Structure paper
タイトル | Mapping Ligand Interactions of Bromodomains BRD4 and ATAD2 with FragLites and PepLites─Halogenated Probes of Druglike and Peptide-like Molecular Interactions. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 65, Page 15416-15432, Year 2022 |
掲載日 | 2021年9月15日 (構造データの登録日) |
![]() | Davison, G. / Martin, M.P. / Turberville, S. / Dormen, S. / Heath, R. / Heptinstall, A.B. / Lawson, M. / Miller, D.C. / Ng, Y.M. / Sanderson, J.N. ...Davison, G. / Martin, M.P. / Turberville, S. / Dormen, S. / Heath, R. / Heptinstall, A.B. / Lawson, M. / Miller, D.C. / Ng, Y.M. / Sanderson, J.N. / Hope, I. / Wood, D.J. / Cano, C. / Endicott, J.A. / Hardcastle, I.R. / Noble, M.E.M. / Waring, M.J. |
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手法 | X線回折 |
解像度 | 0.988 - 2.52 Å |
構造データ | ![]() PDB-7ppx: ![]() PDB-7qu7: ![]() PDB-7quk: ![]() PDB-7qum: ![]() PDB-7qwo: ![]() PDB-7qx1: ![]() PDB-7qxt: ![]() PDB-7qyk: ![]() PDB-7qyl: ![]() PDB-7qzm: ![]() PDB-7qzy: ![]() PDB-7qzz: ![]() PDB-7r00: ![]() PDB-7r05: ![]() PDB-7r0y: ![]() PDB-7z9h: ![]() PDB-7z9i: ![]() PDB-7z9j: ![]() PDB-7z9n: ![]() PDB-7z9o: ![]() PDB-7z9s: ![]() PDB-7z9u: ![]() PDB-7z9w: ![]() PDB-7z9y: ![]() PDB-7za6: ![]() PDB-7za7: ![]() PDB-7za8: ![]() PDB-7za9: ![]() PDB-7zaa: ![]() PDB-7zad: ![]() PDB-7zae: ![]() PDB-7zaj: ![]() PDB-7zaq: ![]() PDB-7zar: ![]() PDB-7zat: ![]() PDB-7ze6: ![]() PDB-7ze7: ![]() PDB-7zef: ![]() PDB-7zen: ![]() PDB-7zfn: ![]() PDB-7zfo: ![]() PDB-7zfs: ![]() PDB-7zft: ![]() PDB-7zfu: ![]() PDB-7zfv: ![]() PDB-7zfy: ![]() PDB-7zfz: ![]() PDB-7zg1: ![]() PDB-7zg2: |
化合物 | ![]() ChemComp-SO4: ![]() ChemComp-CL: ![]() ChemComp-7ZX: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-HH8: ![]() ChemComp-BYZ: ![]() ChemComp-PYZ: ![]() ChemComp-HGQ: ![]() ChemComp-HHQ: ![]() ChemComp-1P8: ![]() ChemComp-IJF: ![]() ChemComp-UU1: ![]() ChemComp-UUS: ![]() ChemComp-V3U: ![]() ChemComp-HHT: ![]() ChemComp-HWC: ![]() ChemComp-HQX: ![]() ChemComp-HNU: ![]() ChemComp-IIV: ![]() ChemComp-IJR: ![]() ChemComp-IIY: ![]() ChemComp-IJ3: ![]() ChemComp-IK3: ![]() ChemComp-IJI: ![]() ChemComp-ARG: ![]() ChemComp-8WS: ![]() ChemComp-GOL: ![]() ChemComp-HEW: ![]() ChemComp-IIS: ![]() ChemComp-IJX: ![]() ChemComp-IJL: ![]() ChemComp-IJO: ![]() ChemComp-3Z7: ![]() ChemComp-IJU: ![]() ChemComp-UUJ: ![]() ChemComp-UUG: ![]() ChemComp-IT4: ![]() ChemComp-IS0: ![]() ChemComp-IS6: ![]() ChemComp-ISK: ![]() ChemComp-IT8: ![]() ChemComp-T9J: |
由来 |
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![]() | TRANSCRIPTION / Transcription regulation / Activator / Hydrolase / Nucleotide-binding / Fragment binding / inhibitor / ATAD2 / FRAGMENT / BROMODOMAIN / FRAGLITE / BRD4 / FragLites / anomalous / Fragment screening |