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-Structure paper
Title | Bidirectional Allosteric Communication between the ATP-Binding Site and the Regulatory PIF Pocket in PDK1 Protein Kinase. |
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Journal, issue, pages | Cell Chem Biol, Vol. 23, Page 1193-1205, Year 2016 |
Publish date | Sep 14, 2016 (structure data deposition date) |
Authors | Schulze, J.O. / Saladino, G. / Busschots, K. / Neimanis, S. / Su, E. / Odadzic, D. / Zeuzem, S. / Hindie, V. / Herbrand, A.K. / Lisa, M.N. ...Schulze, J.O. / Saladino, G. / Busschots, K. / Neimanis, S. / Su, E. / Odadzic, D. / Zeuzem, S. / Hindie, V. / Herbrand, A.K. / Lisa, M.N. / Alzari, P.M. / Gervasio, F.L. / Biondi, R.M. |
External links | Cell Chem Biol / PubMed:27693059 |
Methods | X-ray diffraction |
Resolution | 1.09 - 2.5 Å |
Structure data | PDB-5lvl: PDB-5lvm: PDB-5lvn: PDB-5lvo: PDB-5lvp: |
Chemicals | ChemComp-537: ChemComp-DTD: ChemComp-DMS: ChemComp-HOH: ChemComp-ADE: ChemComp-ADN: ChemComp-CL: ChemComp-ATP: ChemComp-78W: |
Source |
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Keywords | TRANSFERASE / protein kinase / allosteric regulation / small compounds / PIF-pocket |