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Title | Development of new inhibitors against M. tuberculosis CoaBC using a fragment based approach. |
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Journal, issue, pages | To Be Published |
Publish date | Apr 27, 2023 (structure data deposition date) |
![]() | Hess, J. / Mendes, V. / Evans, J.C. / Trapero, A. / Marchetti, C. / Blaszczyk, M. / Bryant, O. / Spry, C. / Coyne, A.G. / Boshoff, H.I.M. ...Hess, J. / Mendes, V. / Evans, J.C. / Trapero, A. / Marchetti, C. / Blaszczyk, M. / Bryant, O. / Spry, C. / Coyne, A.G. / Boshoff, H.I.M. / Barry, C.E. / Mizrahi, V. / Blundell, T.L. / Abell, C. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.993 - 2.84 Å |
Structure data | ![]() PDB-8ow5: ![]() PDB-8owb: ![]() PDB-8owp: ![]() PDB-8owq: ![]() PDB-8owr: |
Chemicals | ![]() ChemComp-CTP: ![]() ChemComp-CA: ![]()
ChemComp-VEO: ![]()
ChemComp-VE6: ![]() ChemComp-HOH: ![]()
ChemComp-W52: ![]() ChemComp-ACT: ![]()
ChemComp-W4X: ![]()
ChemComp-W5E: |
Source |
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![]() | LIGASE / CoaB / CoaBC / Fragment inhibitor |