| タイトル | Disordered DNA-binding motif forms a modulation site for inhibiting the cancer immunotherapy target TREX1. |
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| ジャーナル・号・ページ | Nucleic Acids Res., Vol. 54, Year 2026 |
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| 掲載日 | 2024年11月12日 (構造データの登録日) |
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著者 | Huang, K.W. / Yu Tsai, C. / Wu, C.Y. / Lin, W.C. / Wu, M.T. / Hsu, K.C. / Yu Yang, C. / Chang, I.Y. / Liu, H.M. / Chu, J.W. / Hsiao, Y.Y. |
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リンク | Nucleic Acids Res. / PubMed:41533589 |
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| 手法 | X線回折 |
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| 解像度 | 1.4 - 2 Å |
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| 構造データ | PDB-9kjd: The apo-mTREX1 crystal structure for soaking experiments (Soaking Condition 1) 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-9kje: The apo-mTREX1 crystal structure for soaking experiments (Soaking Condition 2) 手法: X-RAY DIFFRACTION / 解像度: 1.4 Å PDB-9kjf: The apo-mTREX1 crystal structure for soaking experiments (Soaking Condition 3) 手法: X-RAY DIFFRACTION / 解像度: 1.6 Å PDB-9kjg: The mTREX1-NSC 37203 complex structure by co-crystallization (NSC 37203 Complex 1) 手法: X-RAY DIFFRACTION / 解像度: 1.91 Å PDB-9kjh: The mTREX1-NSC 37203 complex structure by soaking in Soaking Condition 1 (NSC 37203 complex 2) 手法: X-RAY DIFFRACTION / 解像度: 1.8 Å PDB-9kji: The mTREX1-NSC 37203 complex structure by co-crystallization (NSC 37203 Complex 3) 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-9kjk: The mTREX1-NSC 37204 complex structure by soaking in Soaking Condition 2 (NSC 37204 complex 1) 手法: X-RAY DIFFRACTION / 解像度: 1.9 Å PDB-9kjl: The mTREX1-NSC 37204 complex structure by soaking in Soaking Condition 3 (NSC 37204 complex 2) 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-9kjm: The mTREX1-NSC 37204 complex structure by soaking in Soaking Condition 1 (NSC 37204 complex 3) 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-9kjn: The mTREX1-NSC 37215 complex structure by co-crystallization (NSC 37215-1 Complex 1) 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-9kjo: The mTREX1-NSC 37215 complex structure by soaking in Soaking Condition 2 (NSC 37215-1 complex 2) 手法: X-RAY DIFFRACTION / 解像度: 2 Å PDB-9kjp: The mTREX1-NSC 37215 complex structure by soaking in Soaking Condition 1 (NSC 37215-2 complex 1) 手法: X-RAY DIFFRACTION / 解像度: 1.9 Å PDB-9kjq: The mTREX1-NSC 37215 complex structure by co-crystallization (NSC 37215-2 Complex 2) 手法: X-RAY DIFFRACTION / 解像度: 1.8 Å PDB-9kjs: The mTREX1-NSC 37215 complex structure by co-crystallization (NSC 37215-2 Complex 3) 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å |
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| 化合物 | ChemComp-EPE: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID / pH緩衝剤*YM
PDB-1l5x: The 2.0-Angstrom resolution crystal structure of a survival protein E (SurE) homolog from Pyrobaculum aerophilum
PDB-1l5z: CRYSTAL STRUCTURE OF THE E121K SUBSTITUTION OF THE RECEIVER DOMAIN OF SINORHIZOBIUM MELILOTI DCTD
PDB-1l50: STRUCTURAL AND THERMODYNAMIC ANALYSIS OF THE PACKING OF TWO ALPHA-HELICES IN BACTERIOPHAGE T4 LYSOZYME
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| 由来 |  mus musculus (ハツカネズミ)
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キーワード | HYDROLASE / TREX1 / Inhibitor / DEDDh exonuclease |
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