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| Title | First Sila-Vitamin D Analogues: Design, Synthesis, Structural Analysis and Biological Activity. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 67, Page 21505-21519, Year 2024 |
| Publish date | Oct 1, 2024 (structure data deposition date) |
Authors | Loureiro, J. / Seoane, S. / Sampaio-Dias, I.E. / Peluso-Iltis, C. / Guiberteau, T. / Brito, B. / Gregorio, C. / Perez-Fernandez, R. / Rochel, N. / Mourino, A. / Rodriguez-Borges, J.E. |
External links | J. Med. Chem. / PubMed:39610329 |
| Methods | X-ray diffraction |
| Resolution | 1.85 - 2.2 Å |
| Structure data | ![]() PDB-9gy8: ![]() PDB-9gya: ![]() PDB-9gyc: ![]() PDB-9gyj: ![]() PDB-9gyk: |
| Chemicals | ![]() PDB-1iqm: ![]() ChemComp-HOH: ![]() ChemComp-ACT: ![]() PDB-1iqq: ![]() PDB-1iqp: ![]() PDB-1iqn: ![]() PDB-1iqo: |
| Source |
|
Keywords | TRANSCRIPTION / VDR complex / agonist / VDR / Complex |
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homo sapiens (human)
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