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Title | Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors. |
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Journal, issue, pages | J. Biol. Chem., Vol. 299, Page 102959-102959, Year 2023 |
Publish date | Sep 12, 2022 (structure data deposition date) |
Authors | Liu, S. / Kormos, B.L. / Knafels, J.D. / Sahasrabudhe, P.V. / Rosado, A. / Sommese, R.F. / Reyes, A.R. / Ward, J. / Roth Flach, R.J. / Wang, X. ...Liu, S. / Kormos, B.L. / Knafels, J.D. / Sahasrabudhe, P.V. / Rosado, A. / Sommese, R.F. / Reyes, A.R. / Ward, J. / Roth Flach, R.J. / Wang, X. / Buzon, L.M. / Reese, M.R. / Bhattacharya, S.K. / Omoto, K. / Filipski, K.J. |
External links | J. Biol. Chem. / PubMed:36717078 |
Methods | X-ray diffraction |
Resolution | 1.85 - 2.047 Å |
Structure data | PDB-8egd: PDB-8egf: PDB-8egq: PDB-8egu: |
Chemicals | ChemComp-ADP: ChemComp-MG: ChemComp-K: ChemComp-SO4: ChemComp-WIH: ChemComp-HOH: ChemComp-WIK: ChemComp-WJK: ChemComp-U35: |
Source |
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Keywords | SIGNALING PROTEIN / Branched-chain ketoacid dehydrogenase / Branched-chain ketoacid dehydrogenase kinase / inhibitors / angiotensin receptor blocker / complex / TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |