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| Title | PCA062, a P-cadherin Targeting Antibody-Drug Conjugate, Displays Potent Antitumor Activity Against P-cadherin-expressing Malignancies. |
|---|---|
| Journal, issue, pages | Mol. Cancer Ther., Vol. 20, Page 1270-1282, Year 2021 |
| Publish date | Jul 17, 2020 (structure data deposition date) |
Authors | Sheng, Q. / D'Alessio, J.A. / Menezes, D.L. / Karim, C. / Tang, Y. / Tam, A. / Clark, S. / Ying, C. / Connor, A. / Mansfield, K.G. ...Sheng, Q. / D'Alessio, J.A. / Menezes, D.L. / Karim, C. / Tang, Y. / Tam, A. / Clark, S. / Ying, C. / Connor, A. / Mansfield, K.G. / Rondeau, J.M. / Ghoddusi, M. / Geyer, F.C. / Gu, J. / McLaughlin, M.E. / Newcombe, R. / Elliot, G. / Tschantz, W.R. / Lehmann, S. / Fanton, C.P. / Miller, K. / Huber, T. / Rendahl, K.G. / Jeffry, U. / Pryer, N.K. / Lees, E. / Kwon, P. / Abraham, J.A. / Damiano, J.S. / Abrams, T.J. |
External links | Mol. Cancer Ther. / PubMed:33879555 |
| Methods | X-ray diffraction |
| Resolution | 1.4 - 2.1 Å |
| Structure data | ![]() PDB-6ztb: ![]() PDB-6ztf: ![]() PDB-6ztr: |
| Chemicals | ![]() ChemComp-CA: ![]() ChemComp-NA: ![]() ChemComp-HOH: |
| Source |
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Keywords | CELL ADHESION / Calcium / Cell Membrane / Glycoprotein / IMMUNE SYSTEM / Immunoglobulin / Fab / Immunoglobulin Cell Adhesion |
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homo sapiens (human)
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