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-Structure paper
Title | Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 4978-4996, Year 2020 |
Publish date | Oct 18, 2019 (structure data deposition date) |
Authors | Ensan, D. / Smil, D. / Zepeda-Velazquez, C.A. / Panagopoulos, D. / Wong, J.F. / Williams, E.P. / Adamson, R. / Bullock, A.N. / Kiyota, T. / Aman, A. ...Ensan, D. / Smil, D. / Zepeda-Velazquez, C.A. / Panagopoulos, D. / Wong, J.F. / Williams, E.P. / Adamson, R. / Bullock, A.N. / Kiyota, T. / Aman, A. / Roberts, O.G. / Edwards, A.M. / O'Meara, J.A. / Isaac, M.B. / Al-Awar, R. |
External links | J. Med. Chem. / PubMed:32369358 |
Methods | X-ray diffraction |
Resolution | 2.09 - 2.56 Å |
Structure data | PDB-6t6d: PDB-8r7g: |
Chemicals | ChemComp-MM8: ChemComp-SO4: ChemComp-HOH:
ChemComp-YEE: |
Source |
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Keywords | SIGNALING PROTEIN / KINASE / BMP / INHIBITOR / SIGNALLING / ALK2 / ACVR1 / M4K2234 |